Sunan samfur:Saukewa: PRL-8-53
OSunan: Methyl 3- (2- (benzylmethylamino) ethyl) benzoate hydrochloride
3- (2-benzylmethylaminoethyl) benzoic acid methyl ester hydrochloride
3- (2- (Methyl (phenylmethyl) amino) ethyl) benzoic acid methyl ester hydrochloride.
Lambar CAS:51352-87-5
Matsayi: 98%
Bayyanar: Farin foda
Ta yaya PRL-8-53 Aiki?
An samo PRL-8-53 daga haɗin benzoic acid da phenylmethylamine.Tsarin sinadarai da aka samu daga haɗuwa da waɗannan mahadi guda biyu yana haifar da wani fili wanda zai iya yin hulɗa tare da masu karɓa na cholinergic, waɗanda ke da hannu wajen daidaita ƙwaƙwalwar ajiya da tsarin ilmantarwa a cikin kwakwalwa.PRL-8-53 kuma an san shi don haɓakawa (ƙara tasirin) dopamine kuma wani ɓangare yana hana masu karɓar serotonin.Dokta Nikolaus Hansl ya yi imanin cewa wannan tasirin tasirin zai iya haifar da canji na ma'auni a cikin tsarin neurotransmitter na CNS kuma ya haifar da ingantaccen aiki na hankali.
An yi nazarin likitancin ɗan adam guda ɗaya kawai wanda aka tsara don kimanta tasirin miyagun ƙwayoyi kuma ya nuna haɓakawa a cikin ƙwaƙwalwar magana, lokacin amsawa na gani da sarrafa motar, musamman a cikin waɗanda suka wuce shekaru 30. Tsofaffi sun fi zama batun ƙwaƙwalwar ajiya. da raguwar fahimi, sabili da haka, ƙwaƙwalwar ajiya da haɓaka haɓakar fahimi suna yin aiki mafi kyau akan su.
Ayyuka RPL-8-53:
Haɓaka hankali na hankali
Ƙarfafa ƙwaƙwalwar ajiya da ƙarfin jingina
Inganta ƙarfin kwakwalwa don magance matsaloli da kare ta daga kowane sinadari ko rauni na jiki
Haɓaka matakin motsawa
Haɓaka sarrafa na'urar kwakwalwa ta cortical/ subcortical
Inganta hangen nesa
Sashi da illa
Bayanan lamba na PRL 8-53 yana nuna kewayon 0.01-4mg/kg na nauyin jiki.Duk da haka, kamar yadda wannan babban kewayon ne, madaidaicin kewayon shine 0.05-1.2 mg/kg.Wannan yana fassara zuwa 3.4mg-81.6mg don mutum 150 da 4.55mg-109mg don mutum 200.A cikin gwajin ɗan adam, ba a sami sakamako mai illa ba;duk da haka, an lura da raguwar ayyukan motsa jiki a cikin beraye da beraye lokacin da aka ba su manyan allurai na PRL 8-53