Ingoa Hua:Tianeptine Hemisulfate Monohydrate
Ētahi atu Ingoa: tianeptinesulfate;
(Thiazepin-11-ylAmino)HeptanoicAcidSemisulfateMonohydrateTianeptineSemisulfateMonohydrate;
7-[(3-Chloro-6,11-dihydro-6-methyl-5,5-dioxidodibenzo[c,f][1,2]thiazepin-11-yl)amino]heptanoicacidsulfatehydrate(2:1:2); Tianeptinehemisulfatemonohydrate(THM);
7-[(3-Chloro-6-methyl-5,5-dioxido-6,11-dihydrodibenzo[c,f][1,2]thiazepin-11-yl)amino]heptanoicacidsulfatehydrate(2:1:2); Tianeptinehemisulfatehydrate;Thiazepin-11-ylAmino)HeptanoicAcidSemisulfate;THM
No CAS:1224690-84-9
Whakatakotoranga: 98.0%
Tae: Te paura karaihe ma me te kakara me te reka
Tūnga GMO: GMO Free
Tapeke: i roto i te 25kgs pahū muka
Rokiroki: Puritia te ipu kia kore e tuwhera ki te waahi makariri, maroke, mawehe atu i te marama kaha
Te Ora: 24 marama mai i te ra o te whakaputanga
Ko te Tianeptine Sulfate/Tianeptine hemisulfate monohydrate he tote pai ake o Tianeptine. Ehara i te hygroscopic no reira he maamaa ake te whakahaere i te paura. I te mea kaore i te rite tonu ki te whakauru me te peia atu i te tinana, ka taea e te tote sulfate te tuku mana ake o te Tianeptine mo nga wa roa. Engari kia toru nga wa ki te horopeta me nga paanga o te tihi tere me nga paanga tere o te heke, ka taea e te tote sulfate kia kotahi te horopeta ki te pupuri i nga taumata plasma i roto i te tinana kia roa ake i te tote konutai. Ko enei ahuatanga kua pai ake ko te Tianeptine Sulfate he taapiri hou.
Ko te Tianeptine Sulfate ehara i te mea he pai noa iho te paanga antidepressant me nga tauhohenga kino i tino iti ake i nga raau taero tricyclic antidepressant tikanga, tata kaore he paanga kino ki te punaha Cardiovascular, toto, ate me nga mahi whatukuhu kaore i whara, kare ano hoki he paanga marie. Ko te Tianeptine ehara i te mea whai hua anake mo te pouri me te neurosis pouri, te waipiro tawhito me te pouri i muri i te waipiro ka whai hua ano hoki. Ko te whakamahi mo te wa roa ka taea te aukati i te hokinga mai
Ko te tianeptine hemisulfate monohydrate, e mohiotia ana ko te tianeptine sulfate, he puhui ahurei i kitea tuatahitia i nga tau 1960, a kua whakamahia nuitia mai i tera wa.
Ko te Tianeptine he antidepressant. Ko te kararehe i te hippocampus pyramidal pūtau nui haere mahorahora, me te whakatere tona mahi i tautāwhi i muri i te whakaora; te whakanui ake i nga cortical me te hippocampalneuron i nga waahi o te 5- serotonin reuptake. Tianeptine me te kore e whai i nga paanga kino: te moe me te mataara; pūnaha cholinergic (kare he tohu anticholinergic); te hiahia tarukino.
Ko te Tianeptine he rongoa rongoa hei whakapai ake i te pouri i roto i ona awhe katoa o te taumahatanga. Ko te rongoa tianeptine e kiia ana he antidepressant tricyclic. He pūhui matū tenei i tapaina na te mea e toru nga mowhiti ngota kei roto.
Pērā i ētahi atu antidepressants tricyclic, ka aukati te tianeptine i te reuptake, te re-absorption ranei, o te serotonin. He neurotransmitter tenei te kawenga mo te oranga o te tangata. Ko te reuptake ka nui ake te waatea o enei matū ki te roro.