Tianeptine Hemisulfate Monohydrate

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Sunan samfur:Tianeptine Hemisulfate Monohydrate

Wani Suna: tianeptinesulfate;

(Thiazepin-11-ylAmino)HeptanoicAcidSemisulfateMonohydrateTianeptineSemisulfateMonohydrate;

7-[(3-Chloro-6,11-dihydro-6-methyl-5,5-dioxidodibenzo[c,f] [1,2] thiazepin-11-yl) amino] heptanoicacidsulfatehydrate (2: 1: 2); Tianeptinehemisulfatemonohydrate (THM);

7-[(3-Chloro-6-methyl-5,5-dioxido-6,11-dihydrodibenzo[c,f] [1,2] thiazepin-11-yl) amino] heptanoicacidsulfatehydrate (2: 1: 2); Tianeptinehemisulfatehydrate;Thiazepin-11-ylAmino)HeptanoicAcidSemisulfate;THM

CAS No:1224690-84-9

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Tianeptine Sulfate/Tianeptine hemisulfate monohydrate shine ingantaccen gishiri na Tianeptine. Ba hygroscopic ba ne don haka sarrafa foda ya fi sauƙi. Tun da yake ba a tsotse shi da sauri kuma yana fitar da shi daga jiki, gishiri sulfate yana ba da damar ƙarin sarrafawar sakin Tianeptine na tsawon lokaci. Maimakon shan kashi sau uku tare da tasirin kololuwa da sauri da faɗuwa da sauri, gishiri sulfate yana ba da damar kashi ɗaya don kula da matakan plasma a cikin jiki fiye da gishirin sodium. Waɗannan ingantattun halaye sun sa Tianeptine Sulfate ya zama ƙari.

Tianeptine Sulfate ba kawai sakamako mai kyau na antidepressant ba da halayen halayen sun kasance ƙasa da na al'ada na antidepressant tricyclic kwayoyi, kusan babu wani tasiri mai tasiri akan tsarin zuciya da jijiyoyin jini, jini, hanta da ayyukan koda ba su ji rauni ba, kuma ba ni da tasiri mai kwantar da hankali. Tianeptine ba wai kawai yana da tasiri ga ɓacin rai da neurosis mai raɗaɗi ba, barasa na yau da kullun da damuwa bayan barasa shima yana da tasiri. Amfani na dogon lokaci zai iya hana sake dawowa

Tianeptine hemisulfate monohydrate, wanda kuma aka sani da tianeptine sulfate, wani fili ne na musamman wanda aka fara gano shi a cikin 1960s kuma tun lokacin ake amfani da shi sosai.

Tianeptine antidepressant ne. Dabbar tana da ƙwayoyin pyramidal na hippocampus sun haɓaka aiki ba tare da bata lokaci ba, kuma an hana haɓaka aikin sa bayan dawowa; karuwa a cikin cortical da hippocampalneurons a wuraren 5- serotonin reuptake. Tianeptine ba tare da bin illa ba: barci da faɗakarwa; tsarin zuciya da jijiyoyin jini; tsarin cholinergic (ba tare da alamun anticholinergic ba); sha'awar miyagun ƙwayoyi.

Tianeptine magani ne na likitanci da ake amfani dashi don inganta ɓacin rai a cikin kowane nau'in tsananinsa. Maganin tianeptine gabaɗaya ana kwatanta shi azaman maganin damuwa na tricyclic. Wannan sinadari ne mai suna saboda yana dauke da zoben atom guda uku.

Kamar sauran tricyclic antidepressants, tianeptine yana toshe sakewa, ko sake sha, na serotonin. Wannan na'ura mai kwakwalwa ce da ke da alhakin jin dadin mutum. Sakamakon sake dawowa yana ƙara samun irin waɗannan abubuwa zuwa kwakwalwa.

Tianeptine hemisulfate monohydrate, wanda kuma aka sani da tianeptine sulfate, wani fili ne na musamman wanda aka fara gano shi a cikin 1960s kuma an yi amfani dashi sosai tun daga lokacin.wanda ke aiki ta hanyar haɓaka sake dawo da serotonin, wani neurotransmitter wanda ke taka muhimmiyar rawa wajen daidaita yanayi da yanayi. . Ta hanyar haɓaka reuptake na serotonin, tianeptine hemisulfate monohydrate yana taimakawa wajen dawo da ma'auni na sinadarai a cikin kwakwalwa, mai yuwuwar rage alamun damuwa. Ɗaya daga cikin keɓancewar sifofin tianeptine hemisulfate monohydrate shine ikonsa na haɓaka neuroplasticity. Neuroplasticity yana nufin ikon kwakwalwa don canzawa da daidaitawa akan lokaci. Bincike ya nuna cewa tianeptine hemisulfate monohydrate yana haɓaka haɓakar sabbin ƙwayoyin cuta kuma yana ƙarfafa haɗin da ke cikin kwakwalwa. Wannan dukiya ta sa ya zama zaɓi mai ban sha'awa don magance damuwa, saboda yana iya ba da fa'idodi na dogon lokaci ban da taimako na alama.

 

Aiki:

Tianeptine sulfate shine maganin damuwa. Dabbobin yana da: Kwayoyin pyramidal na hippocampus sun karu da aiki ba tare da bata lokaci ba, kuma an hana haɓaka aikin sa bayan dawowa; karuwa a cikin cortical da hippocampal neurons a wuraren 5- serotonin reuptake. Tianeptine ba tare da bin illa ba: barci da faɗakarwa; tsarin zuciya da jijiyoyin jini; tsarin cholinergic (ba tare da alamun anticholinergic ba); sha'awar miyagun ƙwayoyi.
Tianeptine Sulfate ba kawai sakamako mai kyau na antidepressant ba da halayen halayen sun kasance ƙasa da na al'ada na antidepressant tricyclic kwayoyi, kusan babu wani tasiri mai tasiri akan tsarin zuciya da jijiyoyin jini, jini, hanta da ayyukan koda ba su ji rauni ba, kuma ba ni da tasiri mai kwantar da hankali. Tianeptine ba wai kawai yana da tasiri ga ɓacin rai da neurosis mai raɗaɗi ba, barasa na yau da kullun da damuwa bayan barasa shima yana da tasiri. Amfani na dogon lokaci zai iya hana sake dawowa.

 

Aikace-aikace:

Tianeptine hemisulfate monohydrate shine zaɓin mai haɓaka reuptake serotonin (SSRE), wanda ke nufin yana haɓaka sake dawo da serotonin a cikin kwakwalwa, ta haka yana haɓaka filastik synaptic da haɓaka yanayi. Yana aiki ta hanyar canza matakan serotonin a cikin kwakwalwa da inganta neuroplasticity. A cikin 'yan shekarun nan, tianeptine hemisulfate monohydrate ya zama sananne a cikin binciken likita, musamman a cikin ci gaba da magungunan maganin damuwa. Kamar yadda ƙarin bincike ya tabbatar da tasirinsa na warkewa, tsammanin aikace-aikacensa yana fitowa a hankali


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