Tianeptine Hemisulfate Monohydrate

Tsanangudzo Pfupi


Product Detail

Product Tags

Product Name:Tianeptine Hemisulfate Monohydrate

Rimwe Zita:tianeptinesulfate;

(Thiazepin-11-ylAmino)HeptanoicAcidSemisulfateMonohydrateTianeptineSemisulfateMonohydrate;

7- [(3-Chloro-6,11-dihydro-6-methyl-5,5-dioxidodibenzo[c,f] [1,2]thiazepin-11-yl) amino]heptanoicacidsulfatehydrate(2:1:2); Tianeptinehemisulfatemonohydrate(THM);

7- [(3-Chloro-6-methyl-5,5-dioxido-6,11-dihydrodibenzo [c,f] [1,2]thiazepin-11-yl) amino]heptanoicacidsulfatehydrate(2:1:2); Tianeptinehemisulfatehydrate;Thiazepin-11-ylAmino)HeptanoicAcidSemisulfate;THM

Nhamba yeCAS:1224690-84-9

Zvinodiwa: 98.0%

Ruvara:White crystal poda ine hunhu hwemunhuwi uye kuravira

GMO Mamiriro:GMO Yemahara

Kurongedza: mune 25kgs fiber zvigubhu

Kuchengeta: Chengetedza mudziyo usina kuvhurwa munzvimbo inotonhorera, yakaoma, Chengetedza kure nechiedza chakasimba

Sherufu Hupenyu: Mwedzi makumi maviri nemana kubva pazuva rekugadzirwa

 

Tianeptine Sulfate/Tianeptine hemisulfate monohydrate inovandudzwa munyu weTianeptine. Haisi hygroscopic saka kubata hupfu kuri nyore kwazvo. Sezvo isiri nyore kunyura uye yakanyungudutswa kubva mumuviri, iyo sulfate munyu inobvumira kudzora kusunungurwa kweTianeptine kwenguva refu. Pane kuti utore katatu nekukasira kwepamusoro mhedzisiro uye nekukurumidza kudonha mhedzisiro, iyo sulfate munyu inobvumira imwe dosi kuchengetedza mazinga eplasma mumuviri kwenguva yakareba kupfuura munyu wesodium. Aya maitiro akavandudzwa anoita kuti Tianeptine Sulfate iwedzere kuwedzera.

Tianeptine Sulfate kwete chete yakanaka antidepressant mhedzisiro uye maitiro akashata aive akanyanya kuderera pane akajairwa antidepressant tricyclic zvinodhaka, zvinenge zvisina mhedzisiro yakaipa pamwoyo, ropa, chiropa uye itsvo mabasa hazvina kukuvadzwa, uye ini handina kudzikamisa maitiro. Tianeptine haisi kungoshanda chete pakuora mwoyo uye kuora mwoyo neurosis, kusingaperi kudhakwa uye kuora mwoyo mushure mekudhakwa kunoshandawo. Kushandiswa kwenguva refu kunogona kudzivirira kudzoka zvakare

Tianeptine hemisulfate monohydrate, inozivikanwawo setianeptine sulfate, isanganiswa yakasarudzika yakatanga kuwanikwa muma1960s uye yakashandiswa zvakanyanya kubva ipapo.

Tianeptine inonzi antidepressant. Mhuka ine hippocampus pyramidal masero yakawedzera kuzviitira basa, uye kukurumidza basa rayo kwakadziviswa mushure mekupora; kuwedzera kwekortical uye hippocampalneurons panzvimbo dze5-serotonin reuptake. Tianeptine pasina kutevera mhedzisiro yakaipa: kurara uye kusvinura; moyo nevascular system; cholinergic system (isina anticholinergic zviratidzo); kuda zvinodhaka.

Tianeptine mushonga wemishonga unoshandiswa kuvandudza kuora mwoyo muzvikamu zvayo zvose zvekuoma. Mushonga wetianeptine unowanzotsanangurwa se tricyclic antidepressant. Uyu musanganiswa wemakemikari wakapihwa zita nekuti une zvindori zvitatu zveatomu.

Kufanana nemamwe tricyclic antidepressants, tianeptine inovhara reuptake, kana kutorazve, ye serotonin. Iyi neurotransmitter inotarisira kunzwa kwemunhu kugara zvakanaka. Reuptake nokudaro inowedzera kuwanikwa kwezvinhu zvakadaro kuuropi.

Tianeptine hemisulfate monohydrate, inozivikanwawo setianeptine sulfate, ikamu rakasiyana rakatanga kuwanikwa muma1960 uye rakashandiswa zvakanyanya kubvira ipapo. . Nekuwedzera serotonin reuptake, tianeptine hemisulfate monohydrate inobatsira kudzoreredza kuenzana kwemakemikari muuropi, zvichigona kuderedza zviratidzo zvekuora mwoyo. Chimwe chezvinhu zvakasarudzika zvetianeptine hemisulfate monohydrate kugona kwayo kuwedzera neuroplasticity. Neuroplasticity inoreva kugona kwehuropi kuchinja uye kugadzirisa nekufamba kwenguva. Tsvagiridzo inoratidza kuti tianeptine hemisulfate monohydrate inosimudzira kukura kwemaneuron matsva uye inosimbisa hukama huripo muuropi. Ichi chivakwa chinoita kuti ive sarudzo inonakidza yekurapa kuora mwoyo, sezvo ichigona kupa mabhenefiti enguva refu mukuwedzera kune zororo rechiratidzo.

 

Basa:

Tianeptine sulfate inonzi antidepressant. Mhuka ine: hippocampus pyramidal masero akawedzera basa rinongoerekana raitika, uye kukurumidza kushanda kwayo kwakadziviswa mushure mekupora; kuwedzera mune cortical uye hippocampal neurons panzvimbo dze5-serotonin reuptake. Tianeptine pasina kutevera migumisiro yakaipa: kurara uye kusvinura; cardiovascular system; cholinergic system (isina anticholinergic zviratidzo); kuda zvinodhaka.
Tianeptine Sulfate kwete chete yakanaka antidepressant mhedzisiro uye maitiro akashata aive akanyanya kuderera pane akajairwa antidepressant tricyclic zvinodhaka, zvinenge zvisina mhedzisiro yakaipa pamwoyo, ropa, chiropa uye itsvo mabasa hazvina kukuvadzwa, uye ini handina kudzikamisa maitiro. Tianeptine haisi kungoshanda chete pakuora mwoyo uye kuora mwoyo neurosis, kusingaperi kudhakwa uye kuora mwoyo mushure mekudhakwa kunoshandawo. Kushandiswa kwenguva refu kunogona kudzivirira kudzoka zvakare.

 

Application:

Tianeptine hemisulfate monohydrate is selective serotonin reuptake enhancer (SSRE), zvinoreva kuti inowedzera kudzokororwa kweserotonin muuropi, nokudaro kuwedzera synaptic plasticity nekuvandudza mafungiro. Inoshanda nekushandura mazinga e serotonin muuropi uye nekusimudzira neuroplasticity. Mumakore achangopfuura, tianeptine hemisulfate monohydrate yakawedzera mukurumbira mukutsvakurudza kwezvokurapa, kunyanya mukugadzirwa kwemishonga inoderedza kuora mwoyo. Sezvo zvidzidzo zvakawanda zvichisimbisa maitiro ayo ekurapa, tarisiro yekushandiswa kwayo iri kubuda zvishoma nezvishoma


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