Product Name:Tianeptine Hemisulfate Monohydrate
Rimwe Zita:tianeptinesulfate;
(Thiazepin-11-ylAmino)HeptanoicAcidSemisulfateMonohydrateTianeptineSemisulfateMonohydrate;
7- [(3-Chloro-6,11-dihydro-6-methyl-5,5-dioxidodibenzo[c,f] [1,2]thiazepin-11-yl) amino]heptanoicacidsulfatehydrate(2:1:2); Tianeptinehemisulfatemonohydrate(THM);
7- [(3-Chloro-6-methyl-5,5-dioxido-6,11-dihydrodibenzo [c,f] [1,2]thiazepin-11-yl) amino]heptanoicacidsulfatehydrate(2:1:2); Tianeptinehemisulfatehydrate;Thiazepin-11-ylAmino)HeptanoicAcidSemisulfate;THM
Nhamba yeCAS:1224690-84-9
Zvinodiwa: 98.0%
Ruvara:White crystal poda ine hunhu hwemunhuwi uye kuravira
GMO Mamiriro:GMO Yemahara
Kurongedza: mune 25kgs fiber zvigubhu
Kuchengeta: Chengetedza mudziyo usina kuvhurwa munzvimbo inotonhorera, yakaoma, Chengetedza kure nechiedza chakasimba
Sherufu Hupenyu: Mwedzi makumi maviri nemana kubva pazuva rekugadzirwa
Tianeptine Sulfate/Tianeptine hemisulfate monohydrate inovandudzwa munyu weTianeptine. Haisi hygroscopic saka kubata hupfu kuri nyore kwazvo. Sezvo isiri nyore kunyura uye yakanyungudutswa kubva mumuviri, iyo sulfate munyu inobvumira kudzora kusunungurwa kweTianeptine kwenguva refu. Pane kuti utore katatu nekukasira kwepamusoro mhedzisiro uye nekukurumidza kudonha mhedzisiro, iyo sulfate munyu inobvumira imwe dosi kuchengetedza mazinga eplasma mumuviri kwenguva yakareba kupfuura munyu wesodium. Aya maitiro akavandudzwa anoita kuti Tianeptine Sulfate iwedzere kuwedzera.
Tianeptine Sulfate kwete chete yakanaka antidepressant mhedzisiro uye maitiro akashata aive akanyanya kuderera pane akajairwa antidepressant tricyclic zvinodhaka, zvinenge zvisina mhedzisiro yakaipa pamwoyo, ropa, chiropa uye itsvo mabasa hazvina kukuvadzwa, uye ini handina kudzikamisa maitiro. Tianeptine haisi kungoshanda chete pakuora mwoyo uye kuora mwoyo neurosis, kusingaperi kudhakwa uye kuora mwoyo mushure mekudhakwa kunoshandawo. Kushandiswa kwenguva refu kunogona kudzivirira kudzoka zvakare
Tianeptine hemisulfate monohydrate, inozivikanwawo setianeptine sulfate, isanganiswa yakasarudzika yakatanga kuwanikwa muma1960s uye yakashandiswa zvakanyanya kubva ipapo.
Tianeptine inonzi antidepressant. Mhuka ine hippocampus pyramidal masero yakawedzera kuzviitira basa, uye kukurumidza basa rayo kwakadziviswa mushure mekupora; kuwedzera kwekortical uye hippocampalneurons panzvimbo dze5-serotonin reuptake. Tianeptine pasina kutevera mhedzisiro yakaipa: kurara uye kusvinura; moyo nevascular system; cholinergic system (isina anticholinergic zviratidzo); kuda zvinodhaka.
Tianeptine mushonga wemishonga unoshandiswa kuvandudza kuora mwoyo muzvikamu zvayo zvose zvekuoma. Mushonga wetianeptine unowanzotsanangurwa se tricyclic antidepressant. Uyu musanganiswa wemakemikari wakapihwa zita nekuti une zvindori zvitatu zveatomu.
Kufanana nemamwe tricyclic antidepressants, tianeptine inovhara reuptake, kana kutorazve, ye serotonin. Iyi neurotransmitter inotarisira kunzwa kwemunhu kugara zvakanaka. Reuptake nokudaro inowedzera kuwanikwa kwezvinhu zvakadaro kuuropi.