Black Atalẹ jade 5.7-Dimethoxyflavone

Apejuwe kukuru:

Atalẹ dudu, iru ọgbin atalẹ kan, dagba ni Asia otutu;O ti pin ni akọkọ ni ariwa ila-oorun Thailand.Ni imọ-jinlẹ, a pe ni Kaempferia parviflora, eyiti a tọka si bi “turmeric dudu” tabi “atalẹ dudu” ni Japan.


  • Iye owo FOB:US $0.5 - 2000 / KG
  • Iye Ibere ​​Min.1 KG
  • Agbara Ipese:10000 KG fun oṣu kan
  • Ibudo:SHANGHAI/BEIJING
  • Awọn ofin sisan:L/C,D/A,D/P,T/T
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  • Alaye ọja

    ọja Tags

    Orukọ ọja:Black Atalẹ jade

    Botanic Orisun:Kaempferia parviflora.L

    CASNìwọ: 21392-57-4

    Orukọ miiran:5.7-Dimethoxyflavone

    Awọn pato: 5.7-Dimethoxyflavone ≥2.5%
    Lapapọ Flavonoids≥10%

    Àwọ̀:eleyi tilulú pẹlu õrùn ti iwa ati itọwo

    GMOIpo: GMO Ọfẹ

    Iṣakojọpọ: ni 25kgs okun ilu

    Ibi ipamọ: Jeki apoti ti a ko ṣii ni itura, aye gbigbẹ, Jeki kuro ni ina to lagbara

    Igbesi aye selifu: awọn oṣu 24 lati ọjọ iṣelọpọ

    5,7-Dimethoxyflavone jẹ ọkan ninu awọn ẹya akọkọ ti Kaempferia parviflora, eyiti o ni egboogi-egbogi isanraju, egboogi-iredodo, ati awọn ipa-egbogi tumo.5,7-Dimethoxyflavone ṣe idiwọ cytochrome P450 (CYP) 3As.5,7-Dimethoxyflavone tun jẹ amuaradagba akàn igbaya ti o munadoko (BCRP) inhibitor.

    Iṣẹ-ṣiṣe inu Vitro:

    Iṣẹ-ṣiṣe trypanocidal vitro ti o dara julọ fun T. brucei rhodesiense ti ṣiṣẹ nipasẹ 7,8-dihydroxyflavone (50% ifọkansi inhibitory [IC50], 68 ng / ml), ti o tẹle 3-hydroxyflavone, rhamnetin, ati 7,8,3′ 4'-tetrahydroxyflavone (IC50s, 0.5 microg / ml) ati catechol (IC50, 0.8 microg / ml)

    Ninu Iṣẹ Vivo:

    5,7-Dimethoxyflavone (10 mg/kg, ẹnu, lẹẹkan lojoojumọ, fun awọn ọjọ 10) le dinku awọn ipele ikosile ti CYP3A11 ati awọn ọlọjẹ CYP3A25 ninu ẹdọ eku [1].

    5,7-Dimethoxyflavone (25 ati 50 mg/kg, oral) le ṣe idiwọ sarcopenia ninu awọn eku agbalagba [3].

    5,7-Dimethoxyflavone (50 mg/kg/d, oral, pípẹ fun ọsẹ 6) le dinku ere iwuwo ati dena ẹdọ ọra ninu awọn eku HFD [5].

    MCE ko tii jẹrisi deede awọn ọna wọnyi.Wọn wa fun itọkasi nikan.

     

     

     

     


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