Orukọ ọja:Black Atalẹ jade
Botanic Orisun:Kaempferia parviflora.L
CASNìwọ: 21392-57-4
Orukọ miiran:5.7-Dimethoxyflavone
Awọn pato: 5.7-Dimethoxyflavone ≥2.5%
Lapapọ Flavonoids≥10%
Àwọ̀:eleyi tilulú pẹlu õrùn ti iwa ati itọwo
GMOIpo: GMO Ọfẹ
Iṣakojọpọ: ni 25kgs okun ilu
Ibi ipamọ: Jeki apoti ti a ko ṣii ni itura, aye gbigbẹ, Jeki kuro ni ina to lagbara
Igbesi aye selifu: awọn oṣu 24 lati ọjọ iṣelọpọ
5,7-Dimethoxyflavone jẹ ọkan ninu awọn ẹya akọkọ ti Kaempferia parviflora, eyiti o ni egboogi-egbogi isanraju, egboogi-iredodo, ati awọn ipa-egbogi tumo.5,7-Dimethoxyflavone ṣe idiwọ cytochrome P450 (CYP) 3As.5,7-Dimethoxyflavone tun jẹ amuaradagba akàn igbaya ti o munadoko (BCRP) inhibitor.
Iṣẹ-ṣiṣe inu Vitro:
Iṣẹ-ṣiṣe trypanocidal vitro ti o dara julọ fun T. brucei rhodesiense ti ṣiṣẹ nipasẹ 7,8-dihydroxyflavone (50% ifọkansi inhibitory [IC50], 68 ng / ml), ti o tẹle 3-hydroxyflavone, rhamnetin, ati 7,8,3′ 4'-tetrahydroxyflavone (IC50s, 0.5 microg / ml) ati catechol (IC50, 0.8 microg / ml)
Ninu Iṣẹ Vivo:
5,7-Dimethoxyflavone (10 mg/kg, ẹnu, lẹẹkan lojoojumọ, fun awọn ọjọ 10) le dinku awọn ipele ikosile ti CYP3A11 ati awọn ọlọjẹ CYP3A25 ninu ẹdọ eku [1].
5,7-Dimethoxyflavone (25 ati 50 mg/kg, oral) le ṣe idiwọ sarcopenia ninu awọn eku agbalagba [3].
5,7-Dimethoxyflavone (50 mg/kg/d, oral, pípẹ fun ọsẹ 6) le dinku ere iwuwo ati dena ẹdọ ọra ninu awọn eku HFD [5].
MCE ko tii jẹrisi deede awọn ọna wọnyi.Wọn wa fun itọkasi nikan.