I-LL-DOPA iwuhlobo lwemvelo lwe-DOPA olusetshenziswa ekwelapheni isifo sika-Parkinson.I-L-DOPA iyisandulela se-dopamine nomkhiqizo we-tyrosine hydroxylase.Okuqondisiwe: I-Dopamine Receptor L-DOPA (L-3,4-dihydroxyphenylalanine) ikhemikhali eyenziwe yaphinde yasetshenziswa njengengxenye ye-biology evamile yabantu, ezinye izilwane nezitshalo.Ezinye izilwane nabantu bakwenza nge-biosynthesis kusuka ku-amino acid L-tyrosine.I-L-DOPA iyisandulela se-neurotransmitters i-dopamine, i-norepinephrine (i-noradrenaline), ne-epinephrine ngokuhlangene eyaziwa ngokuthi ama-catecholamines.I-L-DOPA ingakhiqizwa futhi ngesimo sayo esihlanzekile ithengiswe njengesidakamizwa se-apsychoactive ne-INN levodopa;amagama okuhweba ahlanganisa i-Sinemet, i-Parcopa, i-Atamet, i-Stalevo, i-Madopar, i-Prolopa, njll. Njengesidakamizwa sisetshenziswa ekwelapheni komtholampilo kwe-Parkinson's disease kanye ne-dopamine-responsive dystonia.I-L-DOPA yeqa umgoqo ovikelayo wobuchopho begazi, kuyilapho i-dopamine ngokwayo ayikwazi.Ngakho-ke, i-L-DOPA isetshenziselwa ukwandisa ukugxila kwe-dopamine ekwelapheni isifo sika-Parkinson kanye ne-dopamine-responsive dystonia.Lokhu kwelashwa kwenziwa kwasebenziseka futhi kwafakazelwa ngokomtholampilo nguGeorge Cotzias kanye nozakwabo, abathola ngakho uMklomelo we-Lasker ka-1969.Ukwengeza, i-L-DOPA, ephathwa ngokubambisana ne-DDCI yangaphandle, iye yaphenywa njengendlela yokwelapha engase ibe khona ye-restless leg syndrome.Kodwa-ke, ucwaningo luye lwabonisa "asikho isithombe esicacile sezimpawu ezincishisiwe".I-L-DOPA iyisandulela se-neurotransmitters i-dopamine, i-norepinephrine (noradrenaline), ne-epinephrine (adrenaline) ngokuhlangene eyaziwa ngokuthi ama-catecholamines.
Ngaphandle kwendima yayo yemvelo nebalulekile yebhayoloji, i-L-DOPA iphinde isetshenziswe ekwelashweni komtholampilo kwesifo sika-Parkinson kanye ne-dystonia ephendula i-dopamine.Uma isetshenziswa esimweni sokwenza imithi, igama le-INN elithi 'levodopa' livame ukusetshenziswa.
I-Levodopa iyisengezo sokudla esenzeka ngokwemvelo kanye nesidakamizwa esisebenza ngengqondo esitholakala ezinhlotsheni ezithile zokudla namakhambi (isb, i-Mucuna pruriens, noma ubhontshisi we-velvet), futhi ihlanganiswa kusuka ku-amino acid L-tyrosine emzimbeni nasebuchosheni bezilwane ezincelisayo.
I-Levodopa iyisandulela se-neurotransmitters i-dopamine, i-norepinephrine (i-noradrenaline), ne-epinephrine (adrenaline) eyaziwa ngokuthi i-catecholamines.
Ngaphandle kwendima yayo yemvelo nebalulekile yebhayoloji, i-L-DOPA iphinde isetshenziswe ekwelashweni komtholampilo kwesifo sika-Parkinson kanye ne-dystonia ephendula i-dopamine.Uma isetshenziswa esimweni sokwenza imithi, igama le-INN elithi 'levodopa' livame ukusetshenziswa.
Igama lomkhiqizo: L-dopa 98%
Umthombo Wezitshalo:Mucuna Pruriens Extract
Ingxenye: Imbewu (Yomisiwe, 100% Yemvelo)
Isithako esisebenzayo: Levodopa (L-dopa)
Indlela Yokukhipha: Amanzi/ Utshwala Okusanhlamvu
Ifomu: impushana emhlophe
Ukucaciswa: 5% -99%
Indlela Yokuhlola: I-HPLC
Inombolo ye-CAS: 59-92-7
I-molecular formal: C9H11NO4
Isisindo se-molecule: 197.19
I-Solubility: Ukuncibilika okuhle kusixazululo se-hydro-alcohol
Isimo se-GMO:GMO Mahhala
Ukupakisha: ku-25kgs fiber drums
Isitoreji: Gcina isitsha singavulwa endaweni epholile, eyomile, gwema ukukhanya okuqinile
Impilo Yeshelufu: Izinyanga ezingama-24 kusukela ngosuku lokukhiqiza
Umsebenzi:
- 1 .Iyi-anti-paralysis agitans.Ngokusebenzisa umgoqo wegazi nobuchopho esicutshini sobuchopho, kodwa nge-decarboxylation ye-dopa decarboxylase ibe yi-dopamine, dlala indima.
2. Ngokuthuthumela okubalulekile kanye nokukhubazeka kokukhubazeka kwe-agitans syndrome ye-non-drug immunogenicity, futhi ekukhanyeni okungcono, okunzima, noma abantu abadala abampofu.
3. Khuthaza ukukhula kwemisipha, unciphise isisindo.
4. Ukwanda kwamathambo nokuguqulwa kwe-osteoporosis.
5 .Izithako zokudla.
6. Yelapha i-parkinsonism kanye ne-Pakinsonism syndrome, i-hepatic coma, imisebenzi yehabhu ukuze uthuthukise ukuphaphama kwesiguli, ukuthuthukiswa kwezimpawu.
7 .Khuthaza ukulala, uthuthukise amasosha omzimba.
8 .Ukuncipha komzimba.
9 .Khulisa ukuminyana kwamathambo kanye nokuhlehla kwe-osteoporosis, ukhuphule amandla emisipha, uthuthukise i-libido nokusebenza kocansi.
Isicelo:
I-1.Mucuna Pruriens Extract ingasetshenziswa njengezithako zokudla.
I-2.I-Mucuna Pruriens Extract isetshenziswa njengengxenye ye-adhesives yasolwandle esetshenziswa ukuphila kwe-pelagic.
I-3.I-Mucuna Pruriens Extract ingakhuthaza ukukhula kwemisipha nokwanda kwamathambo kanye nokuguqulwa kwe-osteoporosis.
I-4.I-Mucuna Pruriens Extract ikhulisa ukuminyana kwamathambo kanye nokuguqulwa kwe-osteoporosis, ikhuphule amandla emisipha, ithuthukise i-libido nokusebenza kocansi.
I-5.Ekusetshenzisweni komtholampilo, i-Mucuna Pruriens Extract ilawulwa ekulawuleni isifo sika-Parkinson kanye ne-dopa-responsive dystonia.
6.Ngokuthuthumela okubalulekile kanye nokukhubazeka kokukhubazeka kwe-agitans syndrome ye-non-drug immunogenicity, futhi ekukhanyeni okungcono, okunzima, noma abantu abadala abampofu.
7.Yelapha i-parkinsonism kanye ne-Pakinsonism syndrome, i-hepatic coma, imisebenzi yehabhu ukuthuthukisa ukuphaphama kwesiguli, ukuthuthukiswa kwezimpawu.
I-8.I-Mucuna Pruriens Extract i-anti-paralysis agitans.Ngokusebenzisa umgoqo wegazi nobuchopho esicutshini sobuchopho, kodwa nge-decarboxylation ye-l-dopa decarboxylase ibe yi-dopamine, dlala indima.
I-9.I-Mucuna Pruriens Extract isetshenziselwa ukuzamazama okubalulekile kanye nokukhubazeka kokukhubazeka kwe-agitans syndrome ye-non-drug immunogenicity, futhi ekukhanyeni okungcono, okunzima, noma abantu abadala abampofu.
Olunye ulwazi lwe-TRB | ||
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USFDA,CEP,KOSHER HALAL GMP ISO Izitifiketi | ||
Ikhwalithi Ethembekile | ||
Cishe iminyaka engama-20, ukuthekelisa amazwe nezifunda ezingama-40, amaqoqo angaphezu kuka-2000 akhiqizwa yi-TRB awanazo izinkinga zekhwalithi, inqubo yokuhlanza eyingqayizivele, ukungcola kanye nokulawula ubumsulwa kuhlangana ne-USP, EP kanye ne-CP | ||
Comprehensive Quality System | ||
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▲ Ukulawula idokhumenti | √ | |
▲ Uhlelo Lokuqinisekisa | √ | |
▲ Uhlelo Lokuqeqesha | √ | |
▲ Iphrothokholi Yokucwaninga Kwangaphakathi | √ | |
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▲ Uhlelo Lwezinsiza Zokusebenza | √ | |
▲ Uhlelo Lokulawula Okubalulekile | √ | |
▲ Uhlelo Lokulawula Ukukhiqiza | √ | |
▲ Uhlelo Lokufaka Amalebula Lokupakisha | √ | |
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▲ Uhlelo Lokuqinisekisa Ukuqinisekisa | √ | |
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Lawula Imithombo Yonke Nezinqubo | ||
Ilawule ngokuqinile yonke impahla eluhlaza, izesekeli nezinto zokupakisha. Izinto ezingavuthiwe ezikhethwayo kanye nezinsiza kanye nomphakeli wezinto zokupakisha onenombolo yase-US DMF. |
Abahlinzeki abambalwa bezinto zokusetshenziswa njengesiqinisekiso sokuhlinzekwa.Izikhungo Zokubambisana Eziqinile ezizokwesekaI-Institute of botany/Institution of microbiology/Academy of Science and Technology/University