Aha ngwaahịa:Tianeptine Hemisulfate Monohydrate

Aha ndị ọzọ: tianeptinesulfate;

(Thiazepin-11-ylAmino)HeptanoicAcidSemisulfateMonohydrateTianeptineSemisulfateMonohydrate;

7-[(3-Chloro-6,11-dihydro-6-methyl-5,5-dioxidodibenzo[c,f] [1,2] thiazepin-11-yl) amino] heptanoicacidsulfatehydrate (2: 1: 2); Tianeptinehemisulfatemonohydrate (THM);

7-[(3-Chloro-6-methyl-5,5-dioxido-6,11-dihydrodibenzo[c,f] [1,2] thiazepin-11-yl) amino] heptanoicacidsulfatehydrate (2: 1: 2); Tianeptinehemisulfatehydrate;Thiazepin-11-ylAmino)HeptanoicAcidSemisulfate;THM

CAS Mba:1224690-84-9

Nkọwa: 98.0%

Agba: White crystal ntụ ntụ nwere àgwà na-esi ísì na uto

Ọnọdụ GMO: GMO efu

Mbukota: na 25kgs fiber drum

Nchekwa: Debe akpa na-emegheghị n'ebe dị jụụ, ebe kpọrọ nkụ, zere ọkụ siri ike

Ndụ shelf: ọnwa 24 site na ụbọchị mmepụta

Tianeptine sulfate/Tianeptine hemisulfate monohydrate bụ nnu Tianeptine emelitere. Ọ bụghị hygroscopic ya mere ijikwa ntụ ntụ dị mfe karị. Ebe ọ bụ na ọ naghị etinye aka ngwa ngwa ma na-esi na ahụ pụta, nnu sulfate na-enye ohere maka mwepụta Tianeptine na-achịkwa karịa ogologo oge. Kama ịnwe ọgwụ ugboro atọ na mmetụta kacha elu ngwa ngwa na mmetụta na-ada ngwa ngwa, nnu sulfate na-enye ohere maka otu dose iji nọgide na-enwe ọkwa plasma n'ime ahụ ogologo oge karịa nnu sodium. Njirimara ndị a emelitere na-eme Tianeptine sulfate ka ọ bụrụ mgbakwunye akwụkwọ akụkọ.

Tianeptine sulfate ọ bụghị nanị na mmetụta antidepressant dị mma na mmeghachi omume ọjọọ dị ntakịrị karịa ọgwụ tricyclic antidepressant, ọ fọrọ nke nta ka ọ bụrụ mmetụta ọjọọ na usoro obi, ọbara , imeju na akụrụ arụghị ọrụ, ma ọ bụ enweghị m mmetụta dị jụụ. Tianeptine abụghị naanị dị irè maka ịda mbà n'obi na neurosis nke ịda mbà n'obi, ịṅụbiga mmanya ókè na ịda mbà n'obi mgbe mmanya na-aba n'anya dịkwa irè. Iji ogologo oge eme ihe nwere ike igbochi nlọghachi azụ

Tianeptine hemisulfate monohydrate, nke a makwaara dị ka tianeptine sulfate, bụ ogige pụrụ iche nke achọpụtara na mbụ n'afọ ndị 1960 ma jiri ya mee ihe kemgbe ahụ.

Tianeptine bụ antidepressant. Anụ anụmanụ nwere sel pyramidal hippocampus mụbara spontaneousactivity, na accelerating ya ọrụ amachibidoro mgbe mgbake; mmụba na cortical na hippocampalneurons na saịtị nke 5- serotonin reuptake. Tianeptine na-esoghị mmetụta ọjọọ: ụra na ịmụrụ anya, usoro obi obi; usoro cholinergic (enweghị ihe mgbaàmà anticholinergic); agụụ ọgwụ.

Tianeptine bụ ọgwụ ndenye ọgwụ na-eji eme ka ịda mbà n'obi dịkwuo elu n'ụdị ike ya niile. A na-akọwakarị ọgwụ tianeptine dị ka tricyclic antidepressant. Nke a bụ ngwakọta kemịkalụ aha ya bụ n'ihi na ọ nwere mgbanaka atọ nke atọ.

Dịka antidepressants tricyclic ndị ọzọ, tianeptine na-egbochi iweghachite, ma ọ bụ nnabata ọzọ, nke serotonin. Nke a bụ neurotransmitter na-ahụ maka ọdịmma mmadụ. N'ihi ya, iweghachite ahụ na-abawanye ohere nke ihe ndị dị otú ahụ na ụbụrụ.

Tianeptine hemisulfate monohydrate, nke a makwaara dị ka tianeptine sulfate, bụ ihe pụrụ iche a chọtara na mbụ na 1960 ma jiri ya mee ihe kemgbe ahụ. Nke na-arụ ọrụ site n'ịbawanye reuptake nke serotonin, neurotransmitter nke na-arụ ọrụ dị mkpa n'ịhazi ọnọdụ na ọnọdụ ọnọdụ. . Site n'ịkwalite nnabata serotonin, tianeptine hemisulfate monohydrate na-enyere aka iweghachi nguzozi nke kemịkalụ na ụbụrụ, nwere ike ibelata mgbaàmà nke ịda mbà n'obi. Otu n'ime ihe pụrụ iche nke tianeptine hemisulfate monohydrate bụ ikike ya ịkwalite neuroplasticity. Neuroplasticity na-ezo aka n'ikike ụbụrụ nke ịgbanwe na ime mgbanwe ka oge na-aga. Nnyocha na-egosi na tianeptine hemisulfate monohydrate na-akwalite uto nke neurons ọhụrụ ma na-ewusi njikọ dị na ụbụrụ ike. Ihe onwunwe a na-eme ka ọ bụrụ nhọrọ na-adọrọ mmasị maka ịgwọ ịda mbà n'obi, n'ihi na ọ nwere ike inye uru dị ogologo oge na mgbakwunye na enyemaka mgbaàmà.

Ọrụ:

Tianeptine sulfate bụ antidepressant. Anụmanụ ahụ nwere: mkpụrụ ndụ pyramidal hippocampus mụbara ọrụ onwe ya, na-egbochi ọrụ ya ngwa ngwa mgbe mgbake gasịrị; mmụba na neurons cortical na hippocampal na saịtị nke 5- serotonin reuptake. Tianeptine na-esoghị mmetụta ọjọọ: ụra na ịmụrụ anya; usoro obi obi; usoro cholinergic (enweghị ihe mgbaàmà anticholinergic); agụụ ọgwụ.
Tianeptine sulfate ọ bụghị nanị na mmetụta antidepressant dị mma na mmeghachi omume ọjọọ dị ntakịrị karịa ọgwụ tricyclic antidepressant, ọ fọrọ nke nta ka ọ bụrụ mmetụta ọjọọ na usoro obi, ọbara , imeju na akụrụ arụghị ọrụ, ma ọ bụ enweghị m mmetụta dị jụụ. Tianeptine abụghị naanị dị irè maka ịda mbà n'obi na neurosis nke ịda mbà n'obi, ịṅụbiga mmanya ókè na ịda mbà n'obi mgbe mmanya na-aba n'anya dịkwa irè. Iji ogologo oge eme ihe nwere ike igbochi nlọghachi azụ.

Ngwa:

Tianeptine hemisulfate monohydrate bụ serotonin reuptake enhancer (SSRE), nke pụtara na ọ na-eme ka nnabata nke serotonin dị n'ụbụrụ, si otú ahụ na-amụba synaptic plasticity na imeziwanye ọnọdụ. Ọ na-arụ ọrụ site n'ịgbanwe ọkwa serotonin na ụbụrụ na ịkwalite neuroplasticity. N'afọ ndị na-adịbeghị anya, tianeptine hemisulfate monohydrate aghọwo ihe na-ewu ewu na nyocha ahụike, karịsịa na mmepụta ọgwụ ndị na-egbochi ịda mbà n'obi. Ka ọtụtụ ọmụmụ na-akwado mmetụta ọgwụgwọ ya, atụmanya ngwa ya na-eji nwayọọ nwayọọ na-apụta