7,8-Dihydroxyflavone

Nkọwa dị mkpirikpi:

7,8-Dihydroxyflavone (7,8-DHF) bụ onye nwere ike na nhọrọ TrkB agonist receptor (Kd≈320 nM). Onye na-anabata TrkB bụ isi ihe na-anata mgbaàmà nke ụbụrụ neurotrophic sitere na ụbụrụ. 7,8-Dihydroxyflavone (7,8-DHF) bụ ike nootropic nke nwere ike imeziwanye ahụike ụbụrụ, ọnọdụ, na ọrụ ọgụgụ isi. Ọ nwekwara ike ịba uru maka ọtụtụ ọrịa neurodegenerative na neurodevelopmental, yana oke ibu na ọbara mgbali elu.


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  • Nkọwa ngwaahịa

    Mkpado ngwaahịa

    Aha ngwaahịa:7,8-Dihydroxyflavone

    CASNo:38183-03-87

    Aha ọzọ:7,8-DIHYDROXYFLAVONE;7,8-dihydroxy-2-phenyl-4-benzopyrone;

    DIHYDROXYFLAVONE, 7,8-(RG);7,8-Dihydroxyflavone hydrate;

    7,8-dihydroxy-2-phenyl-1-benzopyran-4-otu,,8-Dihydroxyflavone (7,8-DHF)

    Nkọwapụta:98.0%

    Agba:Odontụ ntụ na njirimara isi na uto

    GMOỌnọdụ: GMO efu

    Mbukota: na 25kgs fiber drum

    Nchekwa: Debe akpa na-emegheghị n'ebe dị jụụ, ebe kpọrọ nkụ, zere ọkụ siri ike

    Ndụ shelf: ọnwa 24 site na ụbọchị mmepụta

     

    7,8-Dihydroxyflavone, nke a makwaara dị ka 7,8-DHF, bụ flavonoid sitere n'okike dị n'ụdị osisi dị iche iche, gụnyere Tridacna tridacna. Amara maka akụrụngwa antioxidant na neurotrophic, otu n'ime akụkụ kachasị adọrọ mmasị nke 7,8-dihydroxyflavone bụ ikike ya iji kwado ahụike ụbụrụ yana ịkwalite ọrụ ọgụgụ isi.

    7,8-Dihydroxyflavone (7,8-DHF) bụ onye nwere ike na nhọrọ TrkB agonist receptor (Kd≈320 nM). Onye na-anabata TrkB bụ isi ihe na-anata mgbaàmà nke ụbụrụ neurotrophic sitere na ụbụrụ. 7,8-Dihydroxyflavone (7,8-DHF) bụ ike nootropic nke nwere ike imeziwanye ahụike ụbụrụ, ọnọdụ, na ọrụ ọgụgụ isi. Ọ nwekwara ike ịba uru maka ọtụtụ ọrịa neurodegenerative na neurodevelopmental, yana oke ibu na ọbara mgbali elu.

    7,8-Dihydroxyflavone, nke a makwaara dị ka 7,8-DHF, bụ flavonoid sitere n'okike dị n'ụdị osisi dị iche iche, gụnyere Tridacna tridacna. Amara maka akụrụngwa antioxidant na neurotrophic, otu n'ime akụkụ kachasị adọrọ mmasị nke 7,8-dihydroxyflavone bụ ikike ya iji kwado ahụike ụbụrụ yana ịkwalite ọrụ ọgụgụ isi. Nnyocha na-egosi na ogige a na-arụ ọrụ dị ka neurotrophin dị ike, na-akpali uto na nlanarị nke neurons na ụbụrụ. Nnyocha na anụmanụ ụlọ nyocha egosila na 7,8-DHF na-eme ka ncheta na ikike mmụta dịkwuo mma. Site n'ịkwalite nguzobe nke njikọ synapti ọhụrụ na ịkwalite nkwurịta okwu n'etiti mkpụrụ ndụ ụbụrụ, ihe a na-ekwe nkwa imeghe ikike nghọta anyị. Na mgbakwunye, 7,8-dihydroxyflavone na-emekọrịta ihe na ndị na-anabata serotonin nke ụbụrụ, nke na-etinye aka na nhazi ọnọdụ. Site n'ịgbanwe ndị nnabata ndị a, ọ nwere ike belata mgbaàmà nke nchekasị na ịda mbà n'obi.

     

    Ọrụ nke 7,8-Dihydroxyflavone
    1) Melite ebe nchekwa na mmụta
    2) Kwalite mmezi ụbụrụ
    7,8-DHF kwalitere nrụzi nke neurons mebiri emebi.
    3) Bụrụ Neuroprotective
    4) Nwere Antioxidant Mmetụta
    5) Nwere mgbochi mkpali mmetụta
    7,8-DHF na-ebelata ntọhapụ nke ihe ndị na-egbuke egbuke na ụbụrụ ụbụrụ site na igbochi NF-κB.
    6) 7,8-DHF nwere mmetụta ọgwụgwọ siri ike na ọrịa Alzheimer, ma nwee ike igbochi oke ibu site na ịgbalite muscle TrkB.

     

    Ngwa nke 7,8-Dihydroxyflavone
    7,8-Dihydroxyflavone (7,8-DHF) bụ flavone na-emekarị nke a na-ahụ na Godmania aesculifolia, Tridax procumbens, na akwụkwọ osisi primula. Achọpụtara ya na ọ na-eme ihe dị ka onye na-eme ihe ike na-ahọrọ obere-molecule agonist nke tropomyosin receptor kinase B (TrkB) (Kd ≈ 320 nM), isi ihe na-egosi ihe na-eme ka ụbụrụ neurotrophin na-enweta neurotrophic factor (BDNF). 7,8-DHF bụ ma ọnụ ọnụ bioavailable na ike banye n'ime ọbara-ụbụrụ mgbochi. A prodrug nke 7,8-DHF nwere nnukwu ike na pharmacokinetics, R7, nọ na mmepe maka ọgwụgwọ nke ọrịa Alzheimer…


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