Tianeptine Hemisulfate Monohydrate

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Tsatanetsatane wa Zamalonda

Zolemba Zamalonda

Dzina lazogulitsa:Tianeptine Hemisulfate Monohydrate

Dzina Lina:tianeptinesulfate;

(Thiazepin-11-ylAmino)HeptanoicAcidSemisulfateMonohydrateTianeptineSemisulfateMonohydrate;

7- [(3-Chloro-6,11-dihydro-6-methyl-5,5-dioxidodibenzo[c,f] [1,2]thiazepin-11-yl) amino]heptanoicacidsulfatehydrate(2:1:2); Tianeptinehemisulfatemonohydrate (THM);

7- [(3-Chloro-6-methyl-5,5-dioxido-6,11-dihydrodibenzo[c,f][1,2]thiazepin-11-yl)amino]heptanoicacidsulfatehydrate(2:1:2); Tianeptinehemisulfatehydrate;Thiazepin-11-ylAmino)HeptanoicAcidSemisulfate;THM

Nambala ya CAS:1224690-84-9

Zofunika: 98.0%

Utoto: ufa wa kristalo woyera wokhala ndi fungo labwino komanso kukoma kwake

Mkhalidwe wa GMO: GMO Yaulere

Kulongedza: mu 25kgs fiber ng'oma

Kusungirako: Sungani chidebe chosatsegulidwa pamalo ozizira, owuma, Khalani kutali ndi kuwala kwamphamvu

Shelf Life: Miyezi 24 kuyambira tsiku lopangidwa

 

Tianeptine Sulfate/Tianeptine hemisulfate monohydrate ndi mchere wabwino wa Tianeptine. Si hygroscopic kotero kuti kugwira ufa kumakhala kosavuta. Popeza sichimatengeka mosavuta ndi kuchotsedwa m'thupi, mchere wa sulphate umalola kuti Tianeptine itulutsidwe kwambiri kwa nthawi yaitali. M'malo mokhala ndi mlingo katatu ndi zotsatira zofulumira kwambiri komanso zotsatira zotsika mofulumira, mchere wa sulphate umalola kuti mlingo umodzi ukhale ndi plasma m'thupi motalika kwambiri kuposa mchere wa sodium. Makhalidwe abwinowa amapangitsa Tianeptine Sulfate kukhala chowonjezera.

Tianeptine sulfate osati zabwino antidepressant zotsatira ndi chokhwima zotsatira anali kwambiri zochepa kuposa ochiritsira antidepressant tricyclic mankhwala, pafupifupi palibe chokhwima pa mtima dongosolo, magazi , chiwindi ndi impso ntchito sizinali zopweteka, kapena ine kukhala bata. Tianeptine sizothandiza kokha kupsinjika maganizo ndi kupsinjika maganizo, kuledzera kosatha ndi kupsinjika maganizo pambuyo pa mowa kumathandizanso. Kugwiritsa ntchito nthawi yayitali kungalepheretse kuyambiranso

Tianeptine hemisulfate monohydrate, yomwe imadziwikanso kuti tianeptine sulfate, ndi gulu lapadera lomwe linapezeka koyamba m'ma 1960 ndipo lakhala likugwiritsidwa ntchito kwambiri kuyambira pamenepo.

Tianeptine ndi antidepressant. Chinyama ali ndi hippocampus piramidi maselo anawonjezera mowiriza ntchito, ndi kufulumizitsa ntchito yake inaletsedwa pambuyo kuchira; kuwonjezeka kwa cortical ndi hippocampalneurons pamasamba a5-serotonin reuptake. Tianeptine popanda zotsatira zoyipa: kugona ndi tcheru;dongosolo lamtima; cholinergic system (popanda zizindikiro za anticholinergic); kulakalaka mankhwala.

Tianeptine ndi mankhwala omwe amagwiritsidwa ntchito popititsa patsogolo kuvutika maganizo m'magulu ake onse. Mankhwala a tianeptine amatchulidwa kuti ndi tricyclic antidepressant. Awa ndi mankhwala opangidwa chifukwa ali ndi ma atomu atatu.

Mofanana ndi mankhwala ena a tricyclic antidepressants, tianeptine imalepheretsa kutenganso, kapena kuyamwanso, kwa serotonin. Ichi ndi neurotransmitter yomwe imapangitsa munthu kukhala ndi moyo wabwino. Kubwerezanso kumawonjezera kupezeka kwa zinthu zotere ku ubongo.

Tianeptine hemisulfate monohydrate, yomwe imadziwikanso kuti tianeptine sulfate, ndi mankhwala apadera omwe anapezeka koyamba m'ma 1960 ndipo akhala akugwiritsidwa ntchito kwambiri kuyambira nthawi imeneyo. . Powonjezera serotonin reuptake, tianeptine hemisulfate monohydrate imathandizira kubwezeretsa mphamvu ya mankhwala muubongo, zomwe zingathe kuchepetsa zizindikiro za kuvutika maganizo. Chimodzi mwazinthu zapadera za tianeptine hemisulfate monohydrate ndi kuthekera kwake kupititsa patsogolo neuroplasticity. Neuroplasticity imatanthawuza kutha kwa ubongo kusintha ndikusintha pakapita nthawi. Kafukufuku akuwonetsa kuti tianeptine hemisulfate monohydrate imathandizira kukula kwa ma neuron atsopano ndikulimbitsa kulumikizana komwe kulipo muubongo. Katunduyu amapangitsa kuti ikhale njira yosangalatsa yochizira kukhumudwa, chifukwa ikhoza kupereka mapindu a nthawi yayitali kuphatikiza pakuchepetsa zizindikiro.

 

Ntchito:

Tianeptine Sulfate ndi antidepressant. Chinyama chili ndi: maselo a hippocampus piramidi adachulukitsa zochitika zokhazokha, ndipo kufulumizitsa ntchito yake kunaletsedwa pambuyo pochira; kuwonjezeka kwa ma cortical ndi hippocampal neurons pamasamba a 5-serotonin reuptake. Tianeptine popanda zotsatira zoyipa: kugona ndi tcheru; mtima dongosolo; cholinergic system (popanda zizindikiro za anticholinergic); kulakalaka mankhwala.
Tianeptine sulfate osati zabwino antidepressant zotsatira ndi chokhwima zotsatira anali kwambiri zochepa kuposa ochiritsira antidepressant tricyclic mankhwala, pafupifupi palibe chokhwima pa mtima dongosolo, magazi , chiwindi ndi impso ntchito sizinali zopweteka, kapena ine ndikukhala bata. Tianeptine sizothandiza kokha kupsinjika maganizo ndi kupsinjika maganizo, kuledzera kosatha ndi kupsinjika maganizo pambuyo pa mowa kumathandizanso. Kugwiritsa ntchito nthawi yayitali kungalepheretse kuyambiranso.

 

Ntchito:

Tianeptine hemisulfate monohydrate ndi serotonin reuptake enhancer (SSRE) yosankha, zomwe zikutanthauza kuti imathandizira kubwezeretsanso kwa serotonin mu ubongo, potero kumawonjezera synaptic plasticity ndikusintha maganizo. Zimagwira ntchito posintha milingo ya serotonin muubongo ndikulimbikitsa neuroplasticity. M'zaka zaposachedwa, tianeptine hemisulfate monohydrate yakhala yotchuka kwambiri mu kafukufuku wamankhwala, makamaka popanga mankhwala osokoneza bongo. Monga momwe kafukufuku wochulukira akutsimikizira zotsatira zake zochiritsira, chiyembekezo chakugwiritsa ntchito kwake chikuwonekera pang'onopang'ono


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