Dzina lazogulitsa:Tianeptine Hemisulfate Monohydrate
Dzina Lina:tianeptinesulfate;
(Thiazepin-11-ylAmino)HeptanoicAcidSemisulfateMonohydrateTianeptineSemisulfateMonohydrate;
7- [(3-Chloro-6,11-dihydro-6-methyl-5,5-dioxidodibenzo[c,f] [1,2]thiazepin-11-yl) amino]heptanoicacidsulfatehydrate(2:1:2); Tianeptinehemisulfatemonohydrate (THM);
7- [(3-Chloro-6-methyl-5,5-dioxido-6,11-dihydrodibenzo[c,f][1,2]thiazepin-11-yl)amino]heptanoicacidsulfatehydrate(2:1:2); Tianeptinehemisulfatehydrate;Thiazepin-11-ylAmino)HeptanoicAcidSemisulfate;THM
Nambala ya CAS:1224690-84-9
Zofunika: 98.0%
Utoto: ufa wa kristalo woyera wokhala ndi fungo labwino komanso kukoma kwake
Mkhalidwe wa GMO: GMO Yaulere
Kulongedza: mu 25kgs fiber ng'oma
Kusungirako: Sungani chidebe chosatsegulidwa pamalo ozizira, owuma, Khalani kutali ndi kuwala kwamphamvu
Shelf Life: Miyezi 24 kuyambira tsiku lopangidwa
Tianeptine Sulfate/Tianeptine hemisulfate monohydrate ndi mchere wabwino wa Tianeptine. Si hygroscopic kotero kuti kugwira ufa kumakhala kosavuta. Popeza sichimatengeka mosavuta ndi kuchotsedwa m'thupi, mchere wa sulphate umalola kuti Tianeptine itulutsidwe kwambiri kwa nthawi yaitali. M'malo mokhala ndi mlingo katatu ndi zotsatira zofulumira kwambiri komanso zotsatira zotsika mofulumira, mchere wa sulphate umalola kuti mlingo umodzi ukhale ndi plasma m'thupi motalika kwambiri kuposa mchere wa sodium. Makhalidwe abwinowa amapangitsa Tianeptine Sulfate kukhala chowonjezera.
Tianeptine sulfate osati zabwino antidepressant zotsatira ndi chokhwima zotsatira anali kwambiri zochepa kuposa ochiritsira antidepressant tricyclic mankhwala, pafupifupi palibe chokhwima pa mtima dongosolo, magazi , chiwindi ndi impso ntchito sizinali zopweteka, kapena ine kukhala bata. Tianeptine sizothandiza kokha kupsinjika maganizo ndi kupsinjika maganizo, kuledzera kosatha ndi kupsinjika maganizo pambuyo pa mowa kumathandizanso. Kugwiritsa ntchito nthawi yayitali kungalepheretse kuyambiranso
Tianeptine hemisulfate monohydrate, yomwe imadziwikanso kuti tianeptine sulfate, ndi gulu lapadera lomwe linapezeka koyamba m'ma 1960 ndipo lakhala likugwiritsidwa ntchito kwambiri kuyambira pamenepo.
Tianeptine ndi antidepressant. Chinyama ali ndi hippocampus piramidi maselo anawonjezera mowiriza ntchito, ndi kufulumizitsa ntchito yake inaletsedwa pambuyo kuchira; kuwonjezeka kwa cortical ndi hippocampalneurons pamasamba a5-serotonin reuptake. Tianeptine popanda zotsatira zoyipa: kugona ndi tcheru;dongosolo lamtima; cholinergic system (popanda zizindikiro za anticholinergic); kulakalaka mankhwala.
Tianeptine ndi mankhwala omwe amagwiritsidwa ntchito popititsa patsogolo kuvutika maganizo m'magulu ake onse. Mankhwala a tianeptine amatchulidwa kuti ndi tricyclic antidepressant. Awa ndi mankhwala opangidwa chifukwa ali ndi ma atomu atatu.
Mofanana ndi mankhwala ena a tricyclic antidepressants, tianeptine imalepheretsa kutenganso, kapena kuyamwanso, kwa serotonin. Ichi ndi neurotransmitter yomwe imapangitsa munthu kukhala ndi moyo wabwino. Kubwerezanso kumawonjezera kupezeka kwa zinthu zotere ku ubongo.