Hesperidin Methyl Chalcone98% nke UV: Nkọwa ngwaahịa zuru oke
1. Okwu Mmalite nke Hesperidin Methyl Chalcone (HMC)
Hesperidin Methyl Chalcone (HMC) bụ ihe methylated sitere na hesperidin, flavonoid na-adịkarị na mkpụrụ citrus dị ka oroma, lemons, na mkpụrụ vaịn. Site na ịdị ọcha nke UV kpebisiri ike nke ≥98%, a na-amata onyinye a maka ọtụtụ uru ya na ahụike vaskụla, nlekọta anụ ahụ, na nchebe antioxidant. Usoro ihe omimi ya bụ C29H36O15 (ihe dị arọ: 624.59 g / mol), a na-ejikwa ya na-acha odo odo na-acha odo odo na ntụ ntụ crystalline nke dị oke hygroscopic na soluble na mmiri, ethanol, na methanol.
2. Nkọwa ngwaahịa
- Nọmba CAS:24292-52-2
- Ịdị ọcha: ≥98% site na nyocha UV
- Ọdịdị: Yellow ka oroma crystalline ntụ ntụ
- Solubility: Nchekwa: Chekwaa n'ebe dị jụụ, kpọrọ nkụ (2-8ºC) pụọ na ìhè na mmiri. Ndụ shelf: afọ 2.
- Na-agbaze kpamkpam na mmiri, ethanol, na methanol.
- Na-agbaze n'otu akụkụ na ethyl acetate.
- Nkwakọ ngwaahịa: 25kg / drum (akpa polyethylene nwere okpukpu abụọ n'ime gbọmgbọm kaadiboodu) .
3. Isi uru na usoro nke ime ihe
3.1 Ahụike akwara na ọbara
HMC na-ewusi capillaries ike site na ibelata permeability na ịkwalite ụda venous, na-eme ka ọ dị irè maka ọgwụgwọ ọnọdụ dị ka ụkọ venous na-adịghị ala ala, hemorrhoid, na veins varicose. Ọmụmụ ụlọ ọgwụ na-egosipụta mmekọrịta ya na yaRuscus aculeatuswepụ na ascorbic acid, nke na-eme ka microcirculation dịkwuo mma ma belata edema.
3.2 Nlekọta akpụkpọ anụ na ngwa akpụkpọ anụ
- Mgbochi ọbara ọbara na mbelata okirikiri gbara ọchịchịrị: HMC na-ebelata ntachi nke capillary n'okpuru anya, na-ebelata mwepu na-acha anụnụ anụnụ na nhịahụ. Ọ bụ isi ihe dị na ude anya adịchaghị mma (dịka ọmụmaatụ,MD Skincare ebuli Lighten Anya ude,Provectin Plus Advanced Eye Cream) .
- Nchedo UV na mgbochi ịka nká: HMC na-egbochi nrụgide oxidative nke UVB, na-egbochi MMP-9 (enzyme na-emebi collagen), ma na-akpali mmepụta filaggrin iji welie ọrụ mgbochi akpụkpọ ahụ.
- Mgbochi Mgbochi na Mmetụta Antioxidant: Site na-egbochi ụzọ NF-κB na IL-6, HMC na-ebelata mbufụt na mmebi oxidative jikọtara na otutu, rosacea, na fotoaging.
3.3 Ọrụ Antioxidant Broad-Spectrum
HMC na-eme ka ụzọ akara Nrf2 rụọ ọrụ, na-akwalite antioxidants endogenous dị ka glutathione na superoxide dismutase. Usoro a na-echebe megide radieshon UV, mmetọ, na nrụgide metabolic.
4. Ngwa na Formulations
4.1 Nutraceuticals
- Usoro onunu ogwu: 30-100 mg / ụbọchị na capsules ma ọ bụ mbadamba maka nkwado venous.
- Usoro ngwakọta: Ọtụtụ mgbe na-ejikọta yaDiosmin,Ascorbic acid, ma ọ bụRuscus wepụmaka nkwalite bioavailability na nrụpụta ọrụ.
4.2 Ihe ịchọ mma na Topicals
- Ntinye uche: 0.5-3% na serums, creams na gels.
- Nhazi igodo:
- Ọgwụ mgbochi ọbara ọbara ọbara: Na-ebelata erythema ihu na uche.
- Ngwaahịa Anya Anya: Ezubere okirikiri gbara ọchịchịrị na nfụkasị (dịka ọmụmaatụ,Gel Anyana menthol maka mmetụta jụrụ oyi).
- Ngwaahịa Nlekọta Sun: Na-arụ ọrụ dị ka ihe nzacha UV (ọnụọgụ absorption na ~ 284 nm) ma na-eme ka Avobenzone guzosie ike na sunscreens.
5. Nkwenye mma na nchekwa
- Nnwale ịdị ọcha: na-agbaso ụkpụrụ pharmacopeial site na iji HPLC na IR spectroscopy.
- Profaịlụ nchekwa: Ọnọdụ nchịkwa: ezute ụkpụrụ FDA nke EU na US maka mgbakwunye nri na ihe ịchọ mma.
- Ndị na-adịghị ewe iwe na usoro akwadoro (LD50> 2000 mg / kg na òké).
- Ọnweghị mutagenicity akọpụtara ma ọ bụ nsi ọmụmụ.
6. Uru Ahịa
- Nnukwu bioavailability: nnabata dị elu ma e jiri ya tụnyere hesperidin nke ala.
- Multifunctionality: Na-eleba anya ma ahụike na ahụike (dịka, ahụike vaskụla + mgbochi ịka nká).
- Nkwado Clinical: Ihe karịrị ọmụmụ nyocha 20 ndị ọgbọ na-akwado ịdị irè ya na nchekwa vaskụla, nguzogide UV, na njikwa mbufụt.
7. Ịtụ na nhazi
- MOQ: 25 kg / drum (nkwakọ ngwaahịa omenala dị).
- Akwụkwọ: COA, MSDS, na data kwụsie ike enyere na arịrịọ .
- Ọrụ OEM: Nhazi ahaziri maka nri nutraceuticals, ịchọ mma, ma ọ bụ ọgwụ.
8. Nkwubi okwu
Hesperidin Methyl Chalcone 98% nke UV bụ ihe dị elu, ihe sayensị na-akwado nke nwere uru egosipụtara maka iguzosi ike n'ezi nke akwara, ahụike anụ ahụ, na nchekwa oxidative. Ọdịiche ya dị na usoro-site na ude anya ruo ihe mgbakwunye venous-na-eme ka ọ bụrụ nhọrọ dabara adaba maka ụdị na-elekwasị anya n'ahịa ndị lekwasịrị anya ahụike na ịma mma.