Lebitso la Sehlahisoa:Tianeptine Hemisulfate Monohydrate
Lebitso le Leng:tianeptinesulfate;
(Thiazepin-11-ylAmino)HeptanoicAcidSemisulfateMonohydrateTianeptineSemisulfateMonohydrate;
7- [(3-Chloro-6,11-dihydro-6-methyl-5,5-dioxidodibenzo [c,f] [1,2]thiazepin-11-yl) amino]heptanoicacidsulfatehydrate (2: 1: 2); Tianeptinehemisulfatemonohydrate(THM);
7- [(3-Chloro-6-methyl-5,5-dioxido-6,11-dihydrodibenzo [c,f] [1,2]thiazepin-11-yl) amino]heptanoicacidsulfatehydrate (2: 1: 2); Tianeptinehemisulfatehydrate;Thiazepin-11-ylAmino)HeptanoicAcidSemisulfate;THM
Nomoro ea CAS:1224690-84-9
Litlhaloso: 98.0%
'Mala: Phofo e tšoeu ea kristale e nang le monko le tatso e ikhethang
Boemo ba GMO:GMO Mahala
Ho paka: ka meqomo ea fiber ea 25kgs
Polokelo: Boloka setshelo se sa buloa sebakeng se phodileng, se omileng, Qoba hole le leseli le matla
Shelf Life: Likhoeli tse 24 ho tloha ka letsatsi la tlhahiso
Tianeptine Sulfate/Tianeptine hemisulfate monohydrate ke letsoai le ntlafetseng la Tianeptine. Ha se hygroscopic kahoo ho sebetsana le phofo ho bonolo haholo. Kaha ha e khone ho kenngoa habonolo le ho tsoa 'meleng, letsoai la sulfate le lumella ho lokolloa ho eketsehileng ho laola Tianeptine ka nako e telele. Ho e-na le ho noa ka makhetlo a mararo ka liphello tse phahameng ka potlako le liphello tse theoha ka potlako, letsoai la sulfate le lumella hore tekanyo e le 'ngoe e boloke boemo ba plasma' meleng nako e telele ho feta letsoai la sodium. Litšobotsi tsena tse ntlafalitsoeng li etsa hore Tianeptine Sulfate e be tlatsetso e ncha.
Tianeptine Sulfate e ne e se feela phello e ntle ea ho tepella maikutlo le liphello tse mpe haholo ho feta lithethefatsi tse tloaelehileng tsa tricyclic, hoo e batlang e se na phello e mpe tsamaisong ea pelo, mali , sebete le liphio ha lia ka tsa utloisoa bohloko, leha e le hore ke na le phello e khutsitseng. Tianeptine ha e sebetse feela bakeng sa ho tepella maikutlong le neurosis e tepeletseng maikutlo, bokhoba ba tahi bo sa foleng le ho tepella maikutlong ka mor'a tai e boetse e sebetsa. Tšebeliso ea nako e telele e ka thibela ho khutla hape
Tianeptine hemisulfate monohydrate, eo hape e tsejoang e le tianeptine sulfate, ke motsoako o ikhethang o qalileng ho fumanoa lilemong tsa bo-1960 'me esale o sebelisoa haholo ho tloha ka nako eo.
Tianeptine ke antidepressant. Phoofolo e na le lisele tsa hippocampus pyramidal e ile ea eketsa ts'ebetso e ikemetseng, 'me ho potlakisa mosebetsi oa eona ho ile ha thibeloa ka mor'a ho hlaphoheloa; keketseho ea cortical le hippocampalneurons libakeng tsa 5-serotonin reuptake. Tianeptine ntle le ho latela liphello tse mpe: ho robala le ho falimeha; tsamaiso ea pelo; tsamaiso ea cholinergic (ntle le matšoao a anticholinergic); takatso ea lithethefatsi.
Tianeptine ke meriana ea ngaka e sebelisoang ho ntlafatsa ho tepella maikutlong ka mefuta eohle ea eona e boima. Hangata meriana ea tianeptine e hlalosoa e le tricyclic antidepressant. Ena ke motsoako oa lik'hemik'hale o bitsoang joalo hobane o na le mehele e meraro ea liathomo.
Joalo ka li-antidepressants tse ling tsa tricyclic, tianeptine e thibela ho khutlisoa, kapa ho monya hape, ea serotonin. Ena ke neurotransmitter e ikarabellang bakeng sa boikutlo ba motho ba boiketlo. Ka lebaka leo, reuptake e eketsa boteng ba lintho tse joalo bokong.