Tianeptine Hemisulfate Monohydrate

Tlhaloso e Khutšoanyane:


Lintlha tsa Sehlahisoa

Li-tag tsa Sehlahisoa

Lebitso la Sehlahisoa:Tianeptine Hemisulfate Monohydrate

Lebitso le Leng:tianeptinesulfate;

(Thiazepin-11-ylAmino)HeptanoicAcidSemisulfateMonohydrateTianeptineSemisulfateMonohydrate;

7- [(3-Chloro-6,11-dihydro-6-methyl-5,5-dioxidodibenzo [c,f] [1,2]thiazepin-11-yl) amino]heptanoicacidsulfatehydrate (2: 1: 2); Tianeptinehemisulfatemonohydrate(THM);

7- [(3-Chloro-6-methyl-5,5-dioxido-6,11-dihydrodibenzo [c,f] [1,2]thiazepin-11-yl) amino]heptanoicacidsulfatehydrate (2: 1: 2); Tianeptinehemisulfatehydrate;Thiazepin-11-ylAmino)HeptanoicAcidSemisulfate;THM

Nomoro ea CAS:1224690-84-9

Litlhaloso: 98.0%

'Mala: Phofo e tšoeu ea kristale e nang le monko le tatso e ikhethang

Boemo ba GMO:GMO Mahala

Ho paka: ka meqomo ea fiber ea 25kgs

Polokelo: Boloka setshelo se sa buloa sebakeng se phodileng, se omileng, Qoba hole le leseli le matla

Shelf Life: Likhoeli tse 24 ho tloha ka letsatsi la tlhahiso

 

Tianeptine Sulfate/Tianeptine hemisulfate monohydrate ke letsoai le ntlafetseng la Tianeptine. Ha se hygroscopic kahoo ho sebetsana le phofo ho bonolo haholo. Kaha ha e khone ho kenngoa habonolo le ho tsoa 'meleng, letsoai la sulfate le lumella ho lokolloa ho eketsehileng ho laola Tianeptine ka nako e telele. Ho e-na le ho noa ka makhetlo a mararo ka liphello tse phahameng ka potlako le liphello tse theoha ka potlako, letsoai la sulfate le lumella hore tekanyo e le 'ngoe e boloke boemo ba plasma' meleng nako e telele ho feta letsoai la sodium. Litšobotsi tsena tse ntlafalitsoeng li etsa hore Tianeptine Sulfate e be tlatsetso e ncha.

Tianeptine Sulfate e ne e se feela phello e ntle ea ho tepella maikutlo le liphello tse mpe haholo ho feta lithethefatsi tse tloaelehileng tsa tricyclic, hoo e batlang e se na phello e mpe tsamaisong ea pelo, mali , sebete le liphio ha lia ka tsa utloisoa bohloko, leha e le hore ke na le phello e khutsitseng. Tianeptine ha e sebetse feela bakeng sa ho tepella maikutlong le neurosis e tepeletseng maikutlo, bokhoba ba tahi bo sa foleng le ho tepella maikutlong ka mor'a tai e boetse e sebetsa. Tšebeliso ea nako e telele e ka thibela ho khutla hape

Tianeptine hemisulfate monohydrate, eo hape e tsejoang e le tianeptine sulfate, ke motsoako o ikhethang o qalileng ho fumanoa lilemong tsa bo-1960 'me esale o sebelisoa haholo ho tloha ka nako eo.

Tianeptine ke antidepressant. Phoofolo e na le lisele tsa hippocampus pyramidal e ile ea eketsa ts'ebetso e ikemetseng, 'me ho potlakisa mosebetsi oa eona ho ile ha thibeloa ka mor'a ho hlaphoheloa; keketseho ea cortical le hippocampalneurons libakeng tsa 5-serotonin reuptake. Tianeptine ntle le ho latela liphello tse mpe: ho robala le ho falimeha; tsamaiso ea pelo; tsamaiso ea cholinergic (ntle le matšoao a anticholinergic); takatso ea lithethefatsi.

Tianeptine ke meriana ea ngaka e sebelisoang ho ntlafatsa ho tepella maikutlong ka mefuta eohle ea eona e boima. Hangata meriana ea tianeptine e hlalosoa e le tricyclic antidepressant. Ena ke motsoako oa lik'hemik'hale o bitsoang joalo hobane o na le mehele e meraro ea liathomo.

Joalo ka li-antidepressants tse ling tsa tricyclic, tianeptine e thibela ho khutlisoa, kapa ho monya hape, ea serotonin. Ena ke neurotransmitter e ikarabellang bakeng sa boikutlo ba motho ba boiketlo. Ka lebaka leo, reuptake e eketsa boteng ba lintho tse joalo bokong.

Tianeptine hemisulfate monohydrate, eo hape e tsejoang e le tianeptine sulfate, ke motsoako o ikhethang o qalileng ho sibolloa lilemong tsa bo-1960 'me o' nile oa sebelisoa haholo ho tloha ka nako eo. . Ka ho ntlafatsa serotonin reuptake, tianeptine hemisulfate monohydrate e thusa ho tsosolosa tekanyo ea lik'hemik'hale bokong, e leng ho ka fokotsang matšoao a ho tepella maikutlong. E 'ngoe ea likarolo tse ikhethang tsa tianeptine hemisulfate monohydrate ke bokhoni ba eona ba ho ntlafatsa neuroplasticity. Neuroplasticity e bolela bokhoni ba boko ba ho fetoha le ho ikamahanya le maemo ha nako e ntse e ea. Lipatlisiso li bontša hore tianeptine hemisulfate monohydrate e khothalletsa kholo ea methapo e mecha le ho matlafatsa likhokahano tse teng bokong. Thepa ena e etsa hore e be khetho e thahasellisang bakeng sa ho phekola ho tepella maikutlong, kaha e ka fana ka melemo ea nako e telele ho phaella ho pholiso ea matšoao.

 

Mosebetsi:

Tianeptine Sulfate ke antidepressant. Phoofolo e na le: lisele tsa hippocampus pyramidal li ile tsa eketsa ts'ebetso e ikemetseng, 'me ho potlakisa mosebetsi oa eona ho ile ha thibeloa ka mor'a ho hlaphoheloa; keketseho ea li-neurons tsa cortical le hippocampal libakeng tsa 5-serotonin reuptake. Tianeptine ntle le ho latela liphello tse mpe: ho robala le ho falimeha; tsamaiso ea methapo ea pelo; tsamaiso ea cholinergic (ntle le matšoao a anticholinergic); takatso ea lithethefatsi.
Tianeptine Sulfate e ne e se feela phello e ntle ea ho tepella maikutlo le liphello tse mpe haholo ho feta lithethefatsi tse tloaelehileng tsa tricyclic, hoo e batlang e se na phello e mpe tsamaisong ea pelo, mali , sebete le liphio ha lia ka tsa utloisoa bohloko, leha e le hore ke na le phello e khutsitseng. Tianeptine ha e sebetse feela bakeng sa ho tepella maikutlong le neurosis e tepeletseng maikutlo, bokhoba ba tahi bo sa foleng le ho tepella maikutlong ka mor'a tai e boetse e sebetsa. Tšebeliso ea nako e telele e ka thibela ho khutlela mokhoeng.

 

Kopo:

Tianeptine hemisulfate monohydrate ke khetho ea serotonin reuptake enhancer (SSRE), e bolelang hore e ntlafatsa ho tsosolosoa ha serotonin bokong, kahoo e eketsa polasetiki ea synaptic le ho ntlafatsa maikutlo. E sebetsa ka ho fetola maemo a serotonin bokong le ho khothaletsa neuroplasticity. Lilemong tsa morao tjena, tianeptine hemisulfate monohydrate e se e tumme haholo lipatlisisong tsa bongaka, haholo-holo ho nts'etsopele ea lithethefatsi tse thibelang ho tepella maikutlo. Ha lithuto tse ntseng li eketseha li tiisa phello ea eona ea phekolo, litebello tsa tšebeliso ea eona li ntse li hlaha butle-butle


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