I-Lemairamin(WGX-50)

Inkcazelo emfutshane:


  • FOB ixabiso:US $ 0.5 - 2000 / KG
  • Min.Ubungakanani boMyalelo:1KG
  • Ukubonelela ngezakhono:I-10000 KG / ngenyanga
  • Izibuko:SHANGHAI/BEIJING
  • Immimiselo yokuhlawula:L/C,D/A,D/P,T/T
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  • Iinkcukacha zeMveliso

    Iithegi zeMveliso

    Igama lemveliso:Lemairamin (WGX-50)

    Elinye Igama:2-Propenamide, N-[2-(3,4-dimethoxyphenyl)ethyl]-3-phenyl-, (2E)-;Lemairamin (WGX-50)

    Inombolo yeCAS:29946-61-0

    Uvavanyo: 98.0%Min

    Umbala: Umhlophe ukuya kumgubo omhlophe

    Ukupakisha:25kg/AMAGUBU

     

    I-Lemairamin okanye i-Wgx50 yinkompawundi yendalo ekhutshwe kwipepile yetshilisi ebonise iziphumo ezithembisayo ekuthinteleni isifo se-Alzheimer. Uphononongo lufumanise ukuba inokuthintela i-Aβ-i-induced neuronal apoptosis, ukunciphisa ubutyhefu be-neuronal calcium, kunye nokunciphisa ukuqokelelwa kwe-Aβ iioligomers kwi-cerebral cortex. Ukongeza, i-wgx50 ibonakaliswe ukuphucula ukusebenza kwengqondo kwiimpuku. Uphando lucebisa ukuba i-wgx50 inamandla okuthintela ukudityaniswa kweeprotheyini phakathi kweeamyloid. Lilonke, i-wgx50 inamandla okuthintela isifo sika-Alzheimer kwaye inokubonelela ngeendlela ezintsha zophuhliso lwamachiza ajolise ku-A.β iioligomers. Ukongezelela, i-WGX-50 ibonisa umsebenzi omkhulu wokuchasana nokuvuvukala, okwenza kube ngumviwa othembisayo wonyango lwezifo ezivuthayo. I-WGX-50 ifunyenwe ibe nemiphumo ebalulekileyo eluswini, njengokunciphisa imibimbi kunye nokuphucula ukuqina kwesikhumba. Ukongeza kwiikhompawundi zendalo ezikhutshwe kwisityalo i-Zanthoxylum bungeanum, okwangoku kukho iikhompawundi ezininzi zokwenziwa ezisetyenziswa kwizicelo ezahlukeneyo kwaye zifaneleke ngakumbi kwimarike.

     

    Umsebenzi:

    1. I-analgesic effect: I-Xanthoxylin ineempawu ze-analgesic kwaye inokunciphisa iimpawu zentlungu. Iyakwazi ukuvuselela ii-receptors zobushushu bomzimba, itshintshe indlela iintlungu ezisasazwa ngayo, kwaye ikhuphe izinto ezidambisa iintlungu ezingapheliyo, ngaloo ndlela inciphisa ukungonwabi okunje ngentloko ebuhlungu kunye nesifo samathambo.
    2. Impembelelo ye-Antibacterial: I-Xanthophyllin ine-antibacterial effect ethile, enokuthintela ukukhula kweebhaktheriya kunye nefungi. Isetyenziswa kakhulu kwishishini lokutya kunye neemveliso zokhathalelo lwempilo ukugcina ukutya kutsha kunye nokwandisa ubomi beshelufu.
    3. Ukukhuthaza ukugaya: I-Xanthoxylum inokukhuthaza ukukhuselwa kweengqungquthela zokugaya, ukunyusa ukukhutshwa kwejusi yesisu kunye ne-saliva, ngaloo ndlela ikhuthaza inkqubo yokugaya ukutya. Inokukhulula iingxaki ze-GI ezifana ne-GI cramps kunye ne-acid reflux.
    4. Umphumo we-Antioxidant: I-Xanthophyllin i-antioxidant enamandla ekwazi ukunciphisa i-radicals yamahhala kunye nokunciphisa umonakalo kwiiseli ezibangelwa uxinzelelo lwe-oxidative. Oku kunceda ukuguga okucothayo, ukukhusela impilo ye-cardiovascular and neurological, kunye nokuthintela ukuphuhliswa kwezifo ezingapheliyo.

     

    Isicelo:

    ILemairamin yikhompawundi ye-amide ekhutshwe kwixolo lesityalo i-Zanthoxylum bungeanum. Okwangoku isetyenziswe njengesongezelelo sokutya, iphinda isebenze njenge-agonist ye-alpha7 nicotinic acetylcholine receptor (α7nAChR), eyanciphisa i-neuroinflammation kwi-Alzheimer's disease.Okwangoku isetyenziswa njengesongezelelo sokutya, iphinda isebenze njenge-agonist ye-alpha7 nicotinic acetylcholine receptor ( α7nAChR), eyanciphisa i-neuroinflammation kwi-Alzheimer's disease, kwaye iphelele i-synthetic.I-Wgx50 ibonise iziphumo ezikhuthazayo kwizifundo zangaphambili, ezibandakanya ukuvimbela i-Aβ-induced neuronal apoptosis, ukunciphisa i-neuronal calcium toxicity, ukunciphisa ukuqokelela kwe-Aβ oligomers kwi-cortex ye-cerebral, kunye nokuphucula ukusebenza kwengqondo kwiigundane.


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