I-Lemairamin(WGX-50)

Incazelo emfushane:


  • Intengo ye-FOB:US $0.5 - 2000 / KG
  • Inani elincane le-oda:1 KG
  • Ikhono Lokuhlinzeka:10000 KG/ngenyanga
  • Imbobo:SHANGHAI/BEIJING
  • Imigomo Yokukhokha:L/C,D/A,D/P,T/T
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  • Imininingwane Yomkhiqizo

    Omaka bomkhiqizo

    Igama Lomkhiqizo:I-Lemairamin (I-WGX-50)

    Elinye Igama:2-Propenamide, N-[2-(3,4-dimethoxyphenyl)ethyl]-3-phenyl-, (2E)-;Lemairamin (I-WGX-50)

    Inombolo ye-CAS:29946-61-0

    Isiqephu: 98.0%Okuncane

    Umbala: Impushana emhlophe ukuya kokumhlophe

    Ukupakisha:25kg/IZIGUbhu

     

    I-Lemairamin noma i-Wgx50 iyinhlanganisela yemvelo ekhishwe kupelepele obonise imiphumela ethembisayo ekuvimbeleni isifo i-Alzheimer's. Ucwaningo luye lwathola ukuthi ingavimbela u-AβI-apoptosis ye-neuronal, inciphisa ubuthi be-neuronal calcium, futhi yehlise ukunqwabelana kwe-Aβ ama-oligomers ku-cortex ye-cerebral. Ngokwengeziwe, i-wgx50 iboniswe ukuthuthukisa ukusebenza kwengqondo kumagundane. Ucwaningo luphakamisa ukuthi i-wgx50 inamandla okuvimbela ukuhlangana kwamaprotheni-namaprotheni phakathi kwama-amyloid molecule. Sekukonke, i-wgx50 inamandla okuvimbela isifo i-Alzheimer's futhi ingase inikeze izindlela ezintsha zokuthuthukiswa kwezidakamizwa eziqondiswe ku-A.β ama-oligomers. Ukwengeza, i-WGX-50 ibonisa umsebenzi obalulekile wokulwa nokuvuvukala, okwenza kube ikhandidethi elithembisayo lokwelapha izifo ezivuthayo. I-WGX-50 itholwe inemiphumela ephawulekayo esikhumbeni, njengokunciphisa imibimbi nokuthuthukisa ukunwebeka kwesikhumba. Ngaphezu kwezinhlanganisela zemvelo ezikhishwe esitshalweni i-Zanthoxylum bungeanum, okwamanje kunezinhlanganisela zokwenziwa ezengeziwe ezisetshenziswa ezinhlelweni ezahlukahlukene futhi ezifaneleke kakhulu emakethe.

     

    Umsebenzi:

    1. Umphumela we-analgesic: I-Xanthoxylin inezindawo zokuqeda ubuhlungu futhi ingadambisa izimpawu zobuhlungu. Ingashukumisa ama-receptors okushisa omzimba, iguqule indlela ubuhlungu obudluliswa ngayo, futhi ikhulule izinto ezidambisa izinhlungu ezingapheli, ngaleyo ndlela yehlise ukungaphatheki kahle okufana nekhanda elibuhlungu nesifo samathambo.
    2. Umphumela we-antibacterial: I-Xanthophyllin inomphumela othile we-antibacterial, ongavimbela ukukhula kwamagciwane kanye nesikhunta. Isetshenziswa kabanzi embonini yokudla kanye nemikhiqizo yokunakekelwa kwezempilo ukuze kugcinwe ukudla kusha futhi kwandise impilo yakho yeshalofu.
    3. Thuthukisa ukugaya: I-Xanthoxylum ingashukumisa ukukhishwa kwezindlala zokugaya, ikhulise ukukhishwa kwejusi yesisu namathe, ngaleyo ndlela ikhuthaze inqubo yokugaya ukudla. Ingase futhi ikhulule izinkinga ze-GI ezifana namajaqamba we-GI kanye ne-acid reflux.
    4. Umphumela we-Antioxidant: I-Xanthophyllin iyi-antioxidant enamandla enganciphisa ama-radicals mahhala futhi inciphise ukulimala kwamaseli okubangelwa ukucindezeleka kwe-oxidative. Lokhu kusiza ukunciphisa ukuguga kwamangqamuzana, kuvikela impilo yenhliziyo nemithambo yegazi, futhi kuvimbele ukuthuthukiswa kwezifo ezingamahlalakhona.

     

    Isicelo:

    I-Lemairamin iyinhlanganisela ye-amide ekhishwe egxolweni lesitshalo se-Zanthoxylum bungeanum. Njengamanje isetshenziswa njengesengezo sokudla, iphinde isebenze njenge-agonist ye-alpha7 nicotinic acetylcholine receptor (α7nAChR), enciphisa i-neuroinflammation ku-Alzheimer's disease.Okwamanje isetshenziswa njengesengezo sokudla, iphinde isebenze njenge-agonist ye-alpha7 nicotinic acetylcholine receptor ( α7nAChR), eyehlisa ukuvuvukala kwe-neuroinflammation ku-Alzheimer's disease, futhi ngokuphelele i-synthetic.I-Wgx50 ibonise imiphumela ekhuthazayo ezifundweni zangaphambi komtholampilo, okuhlanganisa ukuvimbela i-apoptosis ye-neuronal eyenziwe yi-Aβ, ukwehlisa ubuthi be-neuronal calcium, ukwehlisa ukunqwabelana kwama-oligomers e-Aβ ku-cortex yobuchopho, kanye nokuthuthukisa ukusebenza kwengqondo kumagundane.


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