J-147 Ufa

Kufotokozera Kwachidule:

J147 ndi J-147 ndi yamphamvu kwambiri, yogwira ntchito pakamwa komanso yoteteza mitsempha yambiri yomwe imatha kupititsa patsogolo kukumbukira nyama zabwinobwino komanso kupewa kulephera kukumbukira matenda a Alzheimer's (AD) mbewa zosasinthika. Zochita za neurotrophic ndi kukumbukira kukumbukira za J-147 zimagwirizanitsidwa ndi kuwonjezeka kwa milingo ya ubongo yochokera ku neurotrophic factor (BDNF) ndi kufotokozera kwa mapuloteni omvera a BDNF, kupititsa patsogolo kwa LTP, kusungidwa kwa mapuloteni a synaptic, kuchepetsa ma amyloid plaques.


  • Mtengo wa FOB:US $ 0.5 - 2000 / KG
  • Kuchuluka kwa Min.Order:1 kg
  • Kupereka Mphamvu:10000 KG / Mwezi
  • Doko:SHANGHAI/BEIJING
  • Malipiro:L/C,D/A,D/P,T/T
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  • Tsatanetsatane wa Zamalonda

    Zolemba Zamalonda

    Dzina lazogulitsa:J-147 Ufa

    Dzina Lina:2,2,2-Trifluoroacetic acid 1-(2,4-DiMethylphenyl) -2-[(3-Methoxyphenyl)Methylene]hydrazide],J-147j147 ndi

    Nambala ya CAS:1146963-51-0

    Kuyesa: 99.0% Min

    Mtundu: Ufa woyera

    Kunyamula: 25kgs Drums

     

    J-147ndi neuroprotectant yamphamvu kwambiri yomwe imachokera ku curcumin, yomwe imagwira ntchito mu turmeric. Mosiyana ndi curcumin, imadutsa chotchinga cha magazi ndi ubongo bwino kwambiri.

    J-147 ndi yamphamvu kwambiri, yogwira ntchito pakamwa, yoteteza ubongo kuti ipititse patsogolo chidziwitso.
    J-147 imatha kudutsa mosavuta chotchinga muubongo wamagazi (BBB). J-147 ikhoza kuletsa monoamine oxidase B (MAO B) ndi dopamine transporter ndi EC50 mfundo za 1.88 μM ndi 0.649 μM, motsatira. J-147 ili ndi kuthekera kochiza matenda a Alzheimer's

    J-147 ndi neuroprotectant yamphamvu kwambiri pakamwa yomwe imachokera makamaka ku curcumin, yomwe imagwira ntchito mu turmeric. Mosiyana ndi curcumin, imadutsa chotchinga cha magazi ndi ubongo bwino kwambiri. Pakati pawo, J-147 imagwira ntchito pomanga ku ATP synthase. Kuchuluka kwa ATP kumayenderana ndi ukalamba. Kuphatikiza pa kuchuluka kwa ma neurotransmitters NGF ndi BDNF, J-147 imatha kuwongolera izi. Kuphatikiza apo, J-147 imaletsa monoamine oxidase B ndi dopamine transporter. Imalimbikitsa kukula kwa ubongo mwa kuwonjezera kuchuluka kwa mitsempha ya kukula kwa mitsempha (NGF) ndi ubongo-derived neurotrophic factor (BDNF). Chofunika kwambiri, J-147 ikhoza kulimbikitsa kukula kwa maselo atsopano a mitsempha, kupititsa patsogolo luso la ubongo la kuphunzira ndi kukumbukira, komanso kupititsa patsogolo ntchito zamaganizo.

    Ntchito:

    J-147 imatha kudutsa mosavuta chotchinga muubongo wamagazi (BBB).
    J-147 ikhoza kuletsa monoamine oxidase B (MAO B) ndi dopamine transporter ndi EC50 mfundo za 1.88 μM ndi 0.649 μM, motsatira.
    J-147 ili ndi kuthekera kochiza matenda a Alzheimer's (AD).
    J-147 ili ndi kuthekera kochiza matenda a Alzheimer's (AD).

    Ntchito:

    J-147 ndi mankhwala opangira omwe njira yake yayikulu imaphatikizira kukulitsa kwa mitochondrial, potero kukhathamiritsa kupanga mphamvu pama cell. J-147 idapangidwa kuti ipititse patsogolo luso la ubongo lokonzanso ndikudziteteza ku kuwonongeka kobwera chifukwa cha ukalamba mwa kukonza magwiridwe antchito a mitochondrial. Kuphatikiza apo, J-147 imawonetsa anti-yotupa komanso antioxidant katundu, kupititsa patsogolo zotsatira zake za neuroprotective. J-147 ikhoza kulimbikitsa kukula kwa maselo atsopano a mitsempha, kupititsa patsogolo luso la ubongo la kuphunzira ndi kukumbukira, ndi kupititsa patsogolo kugwira ntchito kwa chidziwitso.


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