Igama lemveliso:I-Black Ginger Extract
Umthombo weBhotani:Kaempferia parviflora.L
CASNo: 21392-57-4
Elinye Igama:5.7-Dimethoxyflavone
Iinkcukacha: 5.7-Dimethoxyflavone ≥2.5%
Iyonke iFlavonoids≥10%
Umbala:Mfusaumgubo onevumba elibonakalayo kunye nencasa
GMOIsimo:GMO Mahala
Ukupakisha: kwi-25kgs fiber drums
Ugcino: Gcina isikhongozeli singavulwanga kwindawo epholileyo neyomileyo, Zigcine kude nokukhanya okuqinileyo
Ubomi beShelf: iinyanga ezingama-24 ukusuka kumhla wokuvelisa
I-5,7-Dimethoxyflavone yenye yezinto eziphambili ze-Kaempferia parviflora, ene-anti-obesity, i-anti-inflammatory, kunye ne-anti-tumor effects.I-5,7-Dimethoxyflavone inqanda i-cytochrome P450 (CYP) 3As.I-5,7-Dimethoxyflavone ikwayi-protein esebenzayo yomhlaza wamabele (BCRP) inhibitor.
Umsebenzi we-In Vitro:
Umsebenzi ogqwesileyo we-vitro trypanocidal we-T. brucei rhodesiense wasetyenziswa yi-7,8-dihydroxyflavone (i-50% inhibitory concentration [IC50], 68 ng / ml), ilandelwa yi-3-hydroxyflavone, rhamnetin, kunye ne-7,8,3′, I-4′-tetrahydroxyflavone (IC50s, 0.5 microg / ml) kunye ne-catechol (IC50, 0.8 microg / ml) ?Umsebenzi ochasene ne-T. cruzi wawumodareyitha, kwaye kuphela i-Chrysin dimethylether kunye ne-3-hydroxydaidzein ine-IC50s ngaphantsi kwe-5.0 microg / ml.
KuMsebenzi weVivo:
I-5,7-Dimethoxyflavone (i-10 mg / kg, ngomlomo, kanye ngosuku, kwiintsuku ze-10) inokunciphisa amanqanaba okubonakaliswa kwe-CYP3A11 kunye ne-CYP3A25 iiprotheni kwisibindi seegundane [1].
I-5,7-Dimethoxyflavone (i-25 kunye ne-50 mg / kg, ngomlomo) inokuthintela i-sarcopenia kwiigundane ezikhulileyo [3].
I-5,7-Dimethoxyflavone (i-50 mg / kg / d, ngomlomo, ehlala kwiiveki ze-6) inokunciphisa ubunzima kunye nokuvimbela isibindi esinamafutha kwiigundane ze-HFD [5].
I-MCE ayizange iqinisekise ngokuzimeleyo ukuchaneka kwezi ndlela.Zenzelwe ireferensi kuphela.