Nefiracetam

Inkcazelo emfutshane:

I-Nefiracetam iyingxenye yeklasi yokuphucula ubukrelekrele be-non-border yamachiza, anezakhiwo zeekhemikhali ezahlukeneyo kunye nokuphucula amandla okuqonda kunye nokuthintela umonakalo wokufunda kunye nememori ngemiphumo yabo kwi-cortex ye-cerebral.

I-Nefiracetam yi-nootropic yentsapho ye-racetam. I-Nefiracetam yi-cognitive enhancer ene-IC50 emalunga ne-150-200 μM ye-Ro 5-4864.


  • FOB ixabiso:US $ 0.5 - 2000 / KG
  • Min.Ubungakanani boMyalelo:1KG
  • Ukubonelela ngezakhono:I-10000 KG / ngenyanga
  • Izibuko:SHANGHAI/BEIJING
  • Immimiselo yokuhlawula:L/C,D/A,D/P,T/T
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  • Iinkcukacha zeMveliso

    Iithegi zeMveliso

    Igama lemveliso:Nefiracetam

    Elinye Igama: n-(2,6-dimethylphenyl) -2-oxo-1-pyrrolidineacetamide;NEFIRACETAM;

    2-oxo-1-pyrrolidinylaceticacid,2,6-dimethylanilide;dm9384;n-(2,6-dimethylphenyl) -2-oxo-1-pyrrolidineacetamid;DM-9384,(2-(2-Oxopyrrolidin-1-yl) -N-(2,6-dimethylphenyl)-acetamide);DMMPA

    Inombolo yeCAS:77191-36-7

    Iinkcukacha: 99.0%

    Umbala: Umgubo omhlophe kunye nevumba elibonakalayo kunye nencasa

    Isimo se-GMO:GMO Mahala

    Ukupakisha: kwi-25kgs fiber drums

    Ugcino: Gcina isikhongozeli singavulwanga kwindawo epholileyo neyomileyo, Zigcine kude nokukhanya okuqinileyo

    Ubomi beShelf: iinyanga ezingama-24 ukusuka kumhla wokuvelisa

     

    I-Nefiracetam yeyosapho lwepiracetam, iklasi yeziyobisi ezaziwa ngeempawu zazo zokuphucula ingqondo. I-Nefiracetam yaqala ukwenziwa kwi-1980 yokuqala kwaye yatsala ingqalelo ngokukhawuleza ngenxa yendlela ekhethekileyo yokusebenza kunye nezicelo zonyango ezinokubakho. Le khompawundi ye-racemic kucingelwa ukuba ichaphazela i-neurotransmitters kunye ne-receptors kwingqondo, ekugqibeleni ikhuthaza ukuphuculwa kwezakhono zokuqonda. I-Nefiracetam ngokuyinhloko ichaphazela amanqanaba engqondo ye-acetylcholine, i-neurotransmitter ephambili ejongene nememori, ukufunda kunye nokusebenza kwengqondo. Ngokumodareyitha i-acetylcholine receptors, i-nefiracetam ikhuthaza ukwanda konxibelelwano phakathi kwe-neurons, ngaloo ndlela iphucula iplastiki ye-synaptic kunye nokuphucula ukugcinwa kwememori. Ukongezelela, i-nefiracetam isebenzisana ne-gamma-aminobutyric acid (GABA) i-receptors ukunceda ukulinganisela i-neurotransmitter milieu. Ngokuchaphazela ngokufanelekileyo i-neurotransmitters ye-excitatory kunye ne-inhibitory, i-nefiracetam inceda ukugcina ukusebenza kwengqondo efanelekileyo, ngaloo ndlela iphucula ukugxila, ingqalelo, kunye nokusebenza kwengqondo jikelele.

     

    Imisebenzi:

    I-Nefiracetam iyiyobisi ye-nootropic ye-antidementia yosapho lwe-racetam.

    1. I-Nefiracetam i-nootropic yentsapho ye-racetam.

    2. I-Nefiracetam yi-cognitive enhancer kunye ne-IC50 malunga ne-150-200 μM ye-Ro 5-4864. Le khompawundi isebenze i-L/N-type iziteshi ze-calcium, i-cholinergic, i-monoaminergic kunye ne-GABAergic systems.

    3. I-Nefiracetam ibonisa isenzo esinamandla se-neuroprotective kwi-retinal ischemia-reperfusion model.

     

     

    Isicelo:

    Izongezo zesondlo, isixhasi sesondlo, izongezo zokutya, izongezo zokutya eziheatlh, imathiriyeli ekrwada yamayeza. izongezo zezemidlalo, izongezo zezondlo ezemidlalo
    1. Luhlobo lwezongezo zesondlo.
    2. Inokuphucula i-aerobic metabolism ye-muscle kwaye ikhulise kakhulu amandla emisipha kunye nokunyamezela ukusuka ekudleni kuphela.
    3. Ingasetyenziswa njengesixhasi sesondlo.
    4. Yenye yezona zixhaso zidumileyo nezisebenzayo zezondlo kunye nemveliso eyimfuneko kubakhi bomzimba.
    5. Ikwasetyenziswa ngokubanzi zezinye iimbaleki, njengabadlali bebhola ekhatywayo, abadlali bebasketball njalo njalo..


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