Igama Lomkhiqizo:I-Black Ginger Extract
Umthombo we-Botanic:Kaempferia parviflora.L
I-CASNo:21392-57-4
Elinye Igama:5.7-Dimethoxyflavone
Imininingwane: 5.7-Dimethoxyflavone ≥2.5%
Isamba se-Flavonoids≥10%
Umbala:Okunsomiimpushana enephunga sici nokunambitha
I-GMOIsimo:GMO Mahhala
Ukupakisha: ku-25kgs fiber drums
Isitoreji: Gcina isitsha singavulwa endaweni epholile, eyomile, gwema ukukhanya okuqinile
Impilo Yeshelufu: Izinyanga ezingama-24 kusukela ngosuku lokukhiqiza
I-5,7-Dimethoxyflavone ingenye yezingxenye eziyinhloko ze-Kaempferia parviflora, ene-anti-obesity, anti-inflammatory, ne-anti-tumor effects.I-5,7-Dimethoxyflavone ivimbela i-cytochrome P450 (CYP) 3As.I-5,7-Dimethoxyflavone futhi iyisivimbeli esisebenzayo sokulwa nomdlavuza webele (BCRP).
Umsebenzi we-In Vitro:
Umsebenzi ongcono kakhulu we-in vitro trypanocidal we-T. brucei rhodesiense wenziwa i-7,8-dihydroxyflavone (i-50% inhibitory concentration [IC50], 68 ng/ml), ilandelwa yi-3-hydroxyflavone, rhamnetin, ne-7,8,3′, I-4′-tetrahydroxyflavone (IC50s, 0.5 microg/ml) ne-catechol (IC50, 0.8 microg/ml).?Umsebenzi omelene ne-T. cruzi wawumaphakathi, futhi yi-Chrysin dimethylether kanye ne-3-hydroxydaidzein kuphela eyayinama-IC50s ngaphansi kuka-5.0 microg/ml.
Kumsebenzi we-Vivo:
I-5,7-Dimethoxyflavone (i-10 mg / kg, ngomlomo, kanye ngosuku, izinsuku ezingu-10) inganciphisa amazinga okuveza amaprotheni e-CYP3A11 kanye ne-CYP3A25 esibindi samagundane [1].
I-5,7-Dimethoxyflavone (i-25 ne-50 mg / kg, ngomlomo) ingavimbela i-sarcopenia kumagundane asebekhulile [3].
I-5,7-Dimethoxyflavone (50 mg/kg/d, ngomlomo, ehlala amasonto e-6) inganciphisa ukuzuza kwesisindo futhi ivimbele isibindi esinamafutha kumagundane e-HFD [5].
I-MCE ayizange iqinisekise ngokuzimela ukunemba kwalezi zindlela.Ezethenjwa kuphela.