Dzina lazogulitsa:PRL-8-53
ODzina lake: Methyl 3-(2-(benzylmethylamino)ethyl)benzoate hydrochloride
3-(2-benzylmethylaminoethyl) benzoic acid methyl ester hydrochloride
3-(2-(Methyl(phenylmethyl)amino)ethyl)benzoic acid methylester hydrochloride
Nambala ya CAS :51352-87-5
Chiwerengero: 98%
Maonekedwe: ufa woyera
Kodi PRL-8-53 Imagwira Ntchito Motani?
PRL-8-53 imachokera ku kuphatikiza kwa benzoic acid ndi phenylmethylamine.Kapangidwe ka mankhwala opangidwa kuchokera ku kuphatikiza kwa zinthu ziwirizi kumapangitsa kuti pakhale gulu lomwe lingagwirizane ndi cholinergic receptors, zomwe zimakhudzidwa ndikusintha kukumbukira ndi kuphunzira mkati mwa ubongo.PRL-8-53 imadziwikanso kuti imapangitsa (kuwonjezera zotsatira za) dopamine ndikuletsa pang'ono serotonin receptors.Dr. Nikolaus Hansl ankakhulupirira kuti izi zingapangitse kusintha kwa dongosolo la CNS neurotransmitter ndikupangitsa kuti luntha lizigwira ntchito bwino.
Pakhala pali phunziro limodzi lachipatala laumunthu lomwe linakonzedweratu kuti liwunikire zotsatira za mankhwalawa ndipo linasonyeza kusintha kwa kukumbukira mawu, nthawi yowonekera komanso kuyendetsa galimoto, makamaka kwa anthu opitirira zaka 30. Anthu okalamba amakonda kukumbukira kwambiri. ndi kuchepa kwachidziwitso, chifukwa chake, kukumbukira ndi chidziwitso chowonjezera zowonjezera zimakonda kugwira ntchito bwino pa iwo.
RPL-8-53 Ntchito:
Wonjezerani nzeru zamaganizo
Limbikitsani kukumbukira ndi luso lotsamira
Limbikitsani mphamvu zaubongo kuti muthe kuthana ndi zovuta ndikuziteteza kumankhwala aliwonse kapena kuvulala kwakuthupi
Limbikitsani mulingo wolimbikitsa
Limbikitsani kuwongolera kwa cortical/subcortical brain mechanism
Limbikitsani kuzindikira kwamalingaliro
Mlingo ndi zotsatira zake
Zambiri za patent zomwe zilipo za PRL 8-53 zikuwonetsa kuchuluka kwa 0.01-4mg/kg ya kulemera kwa thupi.Komabe, popeza kuti ndi mtundu waukulu kwambiri, mtundu woyenera ndi 0.05-1.2 mg/kg.Izi zimatanthawuza 3.4mg-81.6mg kwa 150 pounds munthu ndi 4.55mg-109mg pa 200 pounds munthu.M'mayesero aumunthu, palibe zotsatirapo zomwe zinalembedwa;komabe, kuchepa kwa magalimoto kunadziwika mu mbewa ndi makoswe atapatsidwa mlingo waukulu wa PRL 8-53