I-Nefiracetam

Incazelo emfushane:

I-Nefiracetam ingeyeqembu lezidakamizwa ezithuthukisa ukuhlakanipha okungezona emngceleni, ezinezakhiwo zamakhemikhali ezihlukene futhi ezithuthukisa ikhono lokucabanga futhi zivimbele ukulimala kokufunda nenkumbulo ngemiphumela yazo ku-cortex ye-cerebral.

I-Nefiracetam iyi-nootropic yomndeni we-racetam. I-Nefiracetam iyisithuthukisi sokuqonda nge-IC50 cishe engu-150-200 μM ye-Ro 5-4864.


  • Intengo ye-FOB:US $0.5 - 2000 / KG
  • Inani elincane le-oda:1 KG
  • Ikhono Lokuhlinzeka:10000 KG/ngenyanga
  • Imbobo:SHANGHAI/BEIJING
  • Imigomo Yokukhokha:L/C,D/A,D/P,T/T
  • :
  • Imininingwane Yomkhiqizo

    Omaka bomkhiqizo

    Igama Lomkhiqizo:I-Nefiracetam

    Elinye Igama: n-(2,6-dimethylphenyl)-2-oxo-1-pyrrolidineacetamide;NEFIRACETAM;

    2-oxo-1-pyrrolidinylaceticacid,2,6-dimethylanilide;dm9384;n-(2,6-dimethylphenyl) -2-oxo-1-pyrrolidineacetamid;DM-9384,(2-(2-Oxopyrrolidin-1-yl) -N-(2,6-dimethylphenyl)-acetamide);DMMPA

    Inombolo ye-CAS:77191-36-7

    Imininingwane: 99.0%

    Umbala:Impushana emhlophe enephunga nokunambitha

    Isimo se-GMO:GMO Mahhala

    Ukupakisha: ku-25kgs fiber drums

    Isitoreji: Gcina isitsha singavulwa endaweni epholile, eyomile, gwema ukukhanya okuqinile

    Impilo Yeshelufu: Izinyanga ezingama-24 kusukela ngosuku lokukhiqiza

     

    I-Nefiracetam ingeyomndeni we-piracetam, ikilasi lezidakamizwa elaziwa ngezici zazo ezithuthukisa ingqondo. I-Nefiracetam yaqala ukuhlanganiswa ekuqaleni kwawo-1980 futhi yakhanga ngokushesha ngenxa yendlela yayo eyingqayizivele yokusebenza kanye nezinhlelo zokusebenza zokwelapha ezingase zibe khona. Le nhlanganisela ye-racemic kucatshangwa ukuthi ithinta ama-neurotransmitters nama-receptors ebuchosheni, ekugcineni ikhuthaze amakhono okuqonda athuthukisiwe. I-Nefiracetam ngokuyinhloko ithinta amazinga obuchopho e-acetylcholine, i-neurotransmitter eyinhloko ebhekele inkumbulo, ukufunda, nokusebenza kwengqondo. Ngokulungisa ama-acetylcholine receptors, i-nefiracetam ikhuthaza ukuxhumana okwandayo phakathi kwama-neurons, ngaleyo ndlela ithuthukise i-synaptic plasticity futhi ithuthukise ukugcinwa kwenkumbulo. Ukwengeza, i-nefiracetam isebenzisana ne-gamma-aminobutyric acid (GABA) receptors ukusiza ukulinganisa i-neurotransmitter milieu. Ngokuthinta kahle ama-neurotransmitters ajabulisayo futhi avimbelayo, i-nefiracetam isiza ukugcina ukusebenza kahle kobuchopho, ngaleyo ndlela ithuthukise ukugxila, ukunaka, kanye nokusebenza kwengqondo okuphelele.

     

    Imisebenzi:

    I-Nefiracetam iyisidakamizwa se-nootropic antidementia somndeni we-racetam.

    1. I-Nefiracetam iyi-nootropic yomndeni we-racetam.

    2. I-Nefiracetam iyisithuthukisi sokuqonda nge-IC50 cishe ye-150-200 μM ye-Ro 5-4864. Le nhlanganisela yenza iziteshi ze-calcium zohlobo lwe-L/N, i-cholinergic, i-monoaminergic kanye nezinhlelo ze-GABAergic.

    3. I-Nefiracetam ibonisa isenzo esinamandla se-neuroprotective kumodeli ye-retinal ischemia-reperfusion.

     

     

    Isicelo:

    Isengezo sokudla okunomsoco, isithuthukisi somsoco, izithasiselo zokudla, izithasiselo zokudla okunomsoco, izinto ezingavuthiwe zemithi. izithako zezemidlalo, izithasiselo zokudla okunomsoco
    1. Iwuhlobo lwesithasiselo sokudla okunempilo.
    2. Ingathuthukisa i-aerobic metabolism ye-muscle futhi ithuthukise kakhulu amandla emisipha nokukhuthazela okuvela ekudleni kuphela.
    3. Ingasetshenziswa njengesithuthukisi somsoco.
    4. Ingenye yezithako zokudla okunomsoco ezidume kakhulu nezisebenzayo kanye nomkhiqizo obalulekile wabakhi bomzimba.
    5. Ibuye isetshenziswe kabanzi ngabanye abasubathi, njengabadlali bebhola, abadlali bebasketball njalonjalo..


  • Okwedlule:
  • Olandelayo: