Aha ngwaahịa:Oji ginger wepụ
Isi mmalite nke ihe ọkụkụ: Kaempferia parviflora.L
CASNo: 21392-57-4
Aha ọzọ:5.7-Dimethoxyflavone
Nkọwa: 5.7-Dimethoxyflavone ≥2.5%
Mkpokọta flavonoids ≥10%
Agba:Purplentụ ntụ na njirimara isi na uto
GMOỌnọdụ: GMO efu
Mbukota: na 25kgs fiber drum
Nchekwa: Debe akpa na-emegheghị n'ebe dị jụụ, ebe kpọrọ nkụ, zere ọkụ siri ike
Ndụ shelf: ọnwa 24 site na ụbọchị mmepụta
5,7-Dimethoxyflavone bụ otu n'ime ihe ndị bụ isi nke Kaempferia parviflora, nke nwere mgbochi oke ibu, mgbochi mkpali, na mgbochi tumor mmetụta.5,7-Dimethoxyflavone na-egbochi cytochrome P450 (CYP) 3As.5,7-Dimethoxyflavone bụkwa onye na-egbochi ọrịa kansa ara (BCRP).
Ọrụ Vitro:
Ọrụ kacha mma in vitro trypanocidal maka T. brucei rhodesiense bụ nke 7,8-dihydroxyflavone (50% inhibitory concentration [IC50], 68 ng / ml), sochiri 3-hydroxyflavone, rhamnetin, na 7,8,3′, 4'-tetrahydroxyflavone (IC50s, 0.5 microg / ml) na catechol (IC50, 0.8 microg / ml) .? Ọrụ megide T. cruzi bụ agafeghị oke, na naanị Chrysin dimethylether na 3-hydroxydaidzein nwere IC50s na-erughị 5.0 microg / ml.
Na Ọrụ Vivo:
5,7-Dimethoxyflavone (10 mg/kg, ọnụ, otu ugboro kwa ụbọchị, maka ụbọchị 10) nwere ike ibelata ọkwa nkwupụta nke CYP3A11 na CYP3A25 protein na imeju ụmụ oke [1].
5,7-Dimethoxyflavone (25 na 50 mg / kg, ọnụ) nwere ike igbochi sarcopenia na ụmụ oke ndị agadi [3].
5,7-Dimethoxyflavone (50 mg / kg / d, oral, na-adịgide adịgide maka izu 6) nwere ike ibelata ibu ibu ma gbochie imeju abụba na ụmụ oke HFD [5].
MCE akwadobeghị izi ezi nke ụzọ ndị a.Ha bụ naanị maka ntụnye aka.