Amino Tadalafil

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Iinkcukacha zeMveliso

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Igama lemveliso:Amino Tadalafil

Elinye Igama:(6R,12aR)-2-Amino-6-(1,3-benzodioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6] ipyrido[3,4-b]indole-1,4-dion e;AminoTadalafil(6R,12Ar)-2-Amino-6-(1,3-Benzodioxol-5-Yl)-2,3,6,7,12,12A-Hexahydropyrazino[1',2':1,6 ]Pyrido[3,4-B]Indole-1,4 -Dione;(6R,12aR)-2-Amino-6-(benzo[d][1,3]dioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2 ':1,6]pyrido[3,4-b]indol-1,4-dion e;(6R,12aR)-2-amino-6-(benzo[d][1,3]dioxol-5-yl)-2,3,12,12a-tetrahydropyrazino[1',2':1,6 ]pyrido[3,4-b]indole-1,4(6H,7H)-dione

Inombolo yeCAS:385769-84-6

Iinkcukacha: 98.0%

Umbala: Umgubo omhlophe ococekileyo onevumba elibonakalayo kunye nencasa

Isimo se-GMO:GMO Mahala

Ukupakisha: kwi-25kgs fiber drums

Ugcino: Gcina isikhongozeli singavulwanga kwindawo epholileyo neyomileyo, Zigcine kude nokukhanya okuqinileyo

Ubomi beShelf: iinyanga ezingama-24 ukusuka kumhla wokuvelisa

 

I-Amino Tadalafil i-compound efana ne-Tadalafil, kunye namanye amaqela asebenzayo kwisakhiwo sayo athatyathelwa indawo ngamaqela e-amino.I-Amino Tadalafil yinto entsha entsha, i-derivative ye-tadalafil, eyanda kakhulu kwintsimi ye-erectile dysfunction (ED). ). Idibanisa i-amino acid kunye ne-tadalafil, i-FDA-evunyiweyo ye-PDE5 inhibitor eyona nto isetyenziselwa ukuphatha i-ED. Isebenza ngokunyusa ukuhamba kwegazi kwi-penis, ukuvumela amadoda ukuba afezekise kwaye agcine i-erection. Ii-amino acids, kwelinye icala, zidlala indima ebalulekileyo kwimisebenzi eyahlukeneyo yomzimba, kubandakanywa ukuveliswa kweeprotheni, ezizibhloko zokwakha izicubu kunye namalungu. Ukudibanisa kwezi zimbini izithako zenzelwe ukuphucula ukusebenza kweTadalafil ekuphatheni i-ED. Kwaye i-amino Tadalafil yinguqulo ephuculweyo enamandla angaqhelekanga, ephucula ukusebenza kunye nokuguquguquka kwangaphambi kwayo. Ubume bayo beekhemikhali buhlala bufana neTadalafil, kodwa ngokusungulwa kwamaqela e-amino, ifumana iimpawu ezikhethekileyo ezenza ukuba zivelele kwihlabathi lamachiza. Njenge-tadalafil, i-Amino Tadalafil isebenza ngokuvimbela i-phosphodiesterase 5 (PDE5), i-enzyme ejongene nokuphula i-cyclic guanosine monophosphate (cGMP) emzimbeni. I-cGMP yikhompawundi yendalo ekhuthaza ukukhululeka kwemithambo yegazi, ngaloo ndlela inyusa ukuhamba kwegazi. Ngokuthintela i-PDE5, i-amino Tadalafil iqinisekisa ukuqokelela kwe-cGMP, ngaloo ndlela iphucula i-vasodilation kunye nokuphucula ukujikeleza kwegazi. Ukongezelela, abaphandi baye baphonononga amandla ayo okunceda ukunyanga i-benign prostatic hyperplasia (BPH) ngokukhuthaza ukuhamba kwegazi kwi-prostate.

 

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